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There are 208870 results for: content related to: Reversibly Addressing an Allosteric Catalyst In Situ: Catalytic Molecular Tweezers

  1. Reversibly Addressing an Allosteric Catalyst In Situ: Catalytic Molecular Tweezers

    Angewandte Chemie

    Volume 116, Issue 41, October 18, 2004, Pages: 5619–5623, Nathan C. Gianneschi, So-Hye Cho, SonBinh T. Nguyen and Chad A. Mirkin

    Version of Record online : 13 OCT 2004, DOI: 10.1002/ange.200460932

  2. Artificial Allosteric Receptors

    Chemistry - A European Journal

    Volume 19, Issue 20, May 10, 2013, Pages: 6162–6196, Dipl.-Chem. Christopher Kremer and Prof. Dr. Arne Lützen

    Version of Record online : 5 MAR 2013, DOI: 10.1002/chem.201203814

  3. Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands

    Chemistry - A European Journal

    Volume 21, Issue 39, September 21, 2015, Pages: 13598–13608, Dr. Sara Sattin, Dr. Jiahui Tao, Dr. Gerolamo Vettoretti, Dr. Elisabetta Moroni, Dr. Marzia Pennati, Dr. Alessia Lopergolo, Dr. Laura Morelli, Dr. Antonella Bugatti, Dr. Abbey Zuehlke, Dr. Mike Moses, Dr. Thomas Prince, Dr. Toshiki Kijima, Dr. Kristin Beebe, Dr. Marco Rusnati, Dr. Len Neckers, Dr. Nadia Zaffaroni, Prof. David A. Agard, Prof. Anna Bernardi and Dr. Giorgio Colombo

    Version of Record online : 18 AUG 2015, DOI: 10.1002/chem.201502211

  4. A Novel Approach to the Discovery of Small-Molecule Ligands of CDK2

    ChemBioChem

    Volume 13, Issue 14, September 24, 2012, Pages: 2128–2136, Dr. Mathew P. Martin, Riazul Alam, Dr. Stephane Betzi, Donna J. Ingles, Dr. Jin-Yi Zhu and Prof. Ernst Schönbrunn

    Version of Record online : 14 AUG 2012, DOI: 10.1002/cbic.201200316

  5. Synthesis and Application of the First Radioligand Targeting the Allosteric Binding Pocket of Chemokine Receptor CXCR3

    ChemMedChem

    Volume 7, Issue 8, August 2012, Pages: 1481–1489, Viachaslau Bernat, Prof. Dr. Markus R. Heinrich, Paul Baumeister, Prof. Dr. Armin Buschauer and Dr. Nuska Tschammer

    Version of Record online : 11 JUN 2012, DOI: 10.1002/cmdc.201200184

  6. A Random Forest Model for Predicting Allosteric and Functional Sites on Proteins

    Molecular Informatics

    Volume 35, Issue 3-4, April 2016, Pages: 125–135, Ava S.-Y. Chen, Nicholas J. Westwood, Paul Brear, Graeme W. Rogers, Lazaros Mavridis and John B. O. Mitchell

    Version of Record online : 21 JAN 2016, DOI: 10.1002/minf.201500108

  7. Quantification of Allosteric Interactions at G Protein–Coupled Receptors Using Radioligand Binding Assays

    Unit

    Current Protocols in Pharmacology

    1:1.22.1–1.22.41

    Katie Leach, Patrick M. Sexton and Arthur Christopoulos

    Published Online : 1 MAR 2011, DOI: 10.1002/0471141755.ph0122s52

  8. Overview of Receptor Allosterism

    Unit

    Current Protocols in Pharmacology

    1:1.21.1–1.21.34

    Karen J. Gregory, Patrick M. Sexton and Arthur Christopoulos

    Published Online : 1 DEC 2010, DOI: 10.1002/0471141755.ph0121s51

  9. Engineering an Allosteric Binding Site for Aminoglycosides into TEM1-β-Lactamase

    ChemBioChem

    Volume 12, Issue 6, April 11, 2011, Pages: 904–913, Dr. Alexander N. Volkov, Dr. Humberto Barrios, Dr. Pascale Mathonet, Dr. Christine Evrard, Prof. Marcellus Ubbink, Prof. Jean-Paul Declercq, Prof. Patrice Soumillion and Prof. Jacques Fastrez

    Version of Record online : 18 MAR 2011, DOI: 10.1002/cbic.201000568

  10. Structure–Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

    ChemPlusChem

    Volume 79, Issue 11, November 2014, Pages: 1558–1568, Dr. László Juhász, Dr. Gergely Varga, Andrea Sztankovics, Ferenc Béke, Dr. Tibor Docsa, Dr. Attila Kiss-Szikszai, Prof. Dr. Pál Gergely, Dr. Juraj Kóňa, Dr. Igor Tvaroška and Prof. Dr. László Somsák

    Version of Record online : 9 SEP 2014, DOI: 10.1002/cplu.201402181

  11. Discovery of 2-(2-Benzoxazoyl amino)-4-Aryl-5-Cyanopyrimidine as Negative Allosteric Modulators (NAMs) of Metabotropic Glutamate Receptor 5 (mGlu5): From an Artificial Neural Network Virtual Screen to an In Vivo Tool Compound

    ChemMedChem

    Volume 7, Issue 3, March 5, 2012, Pages: 406–414, Dr. Ralf Mueller, Dr. Eric S. Dawson, Prof. Jens Meiler, Dr. Alice L. Rodriguez, Dr. Brian A. Chauder, Brittney S. Bates, Dr. Andrew S. Felts, Jeffrey P. Lamb, Usha N. Menon, Dr. Sataywan B. Jadhav, Dr. Alexander S. Kane, Prof. Dr. Carrie K. Jones, Dr. Karen J. Gregory, Prof. Colleen M. Niswender, Prof. P. Jeffrey Conn, Dr. Christopher M. Olsen, Prof. Danny G. Winder, Prof. Kyle A. Emmitte and Prof. Craig W. Lindsley

    Version of Record online : 20 JAN 2012, DOI: 10.1002/cmdc.201100510

  12. Tetrakisphosphates and Bispyrophosphates of myo-Inositol Derivatives as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Oxygen Release

    ChemMedChem

    Volume 6, Issue 1, January 3, 2011, Pages: 169–180, Prof. Alexandros E. Koumbis, Dr. Carolina D. Duarte, Prof. Claude Nicolau and Prof. Jean-Marie Lehn

    Version of Record online : 10 DEC 2010, DOI: 10.1002/cmdc.201000421

  13. Towards Allosteric Receptors: Adjustment of the Rotation Barrier of 2,2′-Bipyridine Derivatives

    Chemistry - A European Journal

    Volume 15, Issue 11, March 2, 2009, Pages: 2572–2580, Stefan Zahn, Werner Reckien, Barbara Kirchner, Holger Staats, Jens Matthey and Arne Lützen

    Version of Record online : 21 JAN 2009, DOI: 10.1002/chem.200801374

  14. Movements Related to Opening, Closing, and Translocation Functions

    Molecular Devices and Machines - A Journey into the Nano World

    Vincenzo Balzani, Alberto Credi, Margeritha Venturi, Pages: 288–328, 2004

    Published Online : 23 FEB 2004, DOI: 10.1002/3527601600.ch12

  15. Terpy(Pt–salphen)2 Switchable Luminescent Molecular Tweezers

    Chemistry - A European Journal

    Volume 20, Issue 48, November 24, 2014, Pages: 15799–15807, Benjamin Doistau, Arnaud Tron, Dr. Sergey A. Denisov, Dr. Gediminas Jonusauskas, Dr. Nathan D. McClenaghan, Geoffrey Gontard, Dr. Valérie Marvaud, Prof. Dr. Bernold Hasenknopf and Dr. Guillaume Vives

    Version of Record online : 6 OCT 2014, DOI: 10.1002/chem.201404064

  16. Polyphosphates and Pyrophosphates of Hexopyranoses as Allosteric Effectors of Human Hemoglobin: Synthesis, Molecular Recognition, and Effect on Oxygen Release

    ChemMedChem

    Volume 6, Issue 1, January 3, 2011, Pages: 153–168, Prof. Konstantina C. Fylaktakidou, Dr. Carolina D. Duarte, Prof. Alexandros E. Koumbis, Prof. Claude Nicolau and Prof. Jean-Marie Lehn

    Version of Record online : 24 NOV 2010, DOI: 10.1002/cmdc.201000366

  17. In Vivo Structure–Activity Relationship Studies Support Allosteric Targeting of a Dual Specificity Phosphatase

    ChemBioChem

    Volume 15, Issue 10, July 7, 2014, Pages: 1436–1445, Vasiliy N. Korotchenko, Manush Saydmohammed, Laura L. Vollmer, Ahmet Bakan, Kyle Sheetz, Karl T. Debiec, Kristina A. Greene, Christine S. Agliori, Ivet Bahar, Billy W. Day, Andreas Vogt and Michael Tsang

    Version of Record online : 6 JUN 2014, DOI: 10.1002/cbic.201402000

  18. Ligand-Biased and Probe-Dependent Modulation of Chemokine Receptor CXCR3 Signaling by Negative Allosteric Modulators

    ChemMedChem

    Volume 10, Issue 3, March 2015, Pages: 566–574, Dr. Viachaslau Bernat, Regine Brox, Prof. Dr. Markus R. Heinrich, Dr. Yves P. Auberson and Dr. Nuska Tschammer

    Version of Record online : 5 FEB 2015, DOI: 10.1002/cmdc.201402507

  19. An Allosteric Synthetic Catalyst: Metal Ions Tune the Activity of an Artificial Phosphodiesterase

    Chemistry - A European Journal

    Volume 7, Issue 6, March 16, 2001, Pages: 1221–1231, Igor O. Fritsky, Reina Ott, Hans Pritzkow and Roland Krämer

    Version of Record online : 8 MAR 2001, DOI: 10.1002/1521-3765(20010316)7:6<1221::AID-CHEM1221>3.0.CO;2-T

  20. Synthesis, SAR and Unanticipated Pharmacological Profiles of Analogues of the mGluR5 Ago-potentiator ADX-47273

    ChemMedChem

    Volume 4, Issue 4, April 17, 2009, Pages: 505–511, Darren W. Engers, Alice L. Rodriguez, Richard Williams, Alexis S. Hammond, Daryl Venable, Oluwatomi Oluwatola, Gary A. Sulikowski, P. Jeffrey Conn and Craig W. Lindsley

    Version of Record online : 5 FEB 2009, DOI: 10.1002/cmdc.200800357