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There are 379050 results for: content related to: Fine Tuning the Inhibition Profile of Cyclosporine A by Derivatization of the MeBmt Residue

  1. Design and Synthesis of Conformationally Constrained Cyclophilin Inhibitors Showing a Cyclosporin-A Phenotype in C. elegans


    Volume 12, Issue 5, March 21, 2011, Pages: 802–810, Dr. Colin J. Dunsmore , Dr. Kirk J. Malone , Dr. Kevin R. Bailey , Dr. Martin A. Wear, Dr. Hannah Florance, Dr. Sally Shirran , Dr. Perdita E. Barran, Prof. Antony P. Page, Prof. Malcolm D. Walkinshaw and Prof. Nicholas J. Turner 

    Article first published online : 17 FEB 2011, DOI: 10.1002/cbic.201000413

  2. Focused Directed Evolution of Pentaerythritol Tetranitrate Reductase by Using Automated Anaerobic Kinetic Screening of Site-Saturated Libraries


    Volume 11, Issue 17, November 22, 2010, Pages: 2433–2447, Martyn E. Hulley, Dr. Helen S. Toogood, Dr. Anna Fryszkowska, Dr. David Mansell, Prof. Gill M. Stephens, Dr. John M. Gardiner and Prof. Nigel S. Scrutton

    Article first published online : 9 NOV 2010, DOI: 10.1002/cbic.201000527

  3. Cytotoxic Fatty Acid Amides from Xenorhabdus


    Volume 12, Issue 13, September 5, 2011, Pages: 2011–2015, Anna Proschak, Katharina Schultz, Jennifer Herrmann, Dr. Andrea J. Dowling, Dr. Alexander O. Brachmann, Prof. Dr. Richard ffrench-Constant, Prof. Dr. Rolf Müller and Prof. Dr. Helge B. Bode

    Article first published online : 12 JUL 2011, DOI: 10.1002/cbic.201100223

  4. Effects of Single Genetic Damage in Carbohydrate-Recognizing Proteins in Mouse Serum N-Glycan Profile Revealed by Simple Glycotyping Analysis


    Volume 13, Issue 3, February 13, 2012, Pages: 451–464, Maho Amano, Ryo Hashimoto and Shin-Ichiro Nishimura

    Article first published online : 24 JAN 2012, DOI: 10.1002/cbic.201100595

  5. Carbohydrate–PNA and Aptamer–PNA Conjugates for the Spatial Screening of Lectins and Lectin Assemblies


    Volume 14, Issue 2, January 21, 2013, Pages: 236–250, Christian Scheibe, Dr. Stefanie Wedepohl, Sebastian B. Riese, Dr. Jens Dernedde and Prof. Dr. Oliver Seitz

    Article first published online : 4 JAN 2013, DOI: 10.1002/cbic.201200618

  6. Kinetics Studies on the Inhibition Mechanism of Pancreatic α-Amylase by Glycoconjugated 1H-1,2,3-Triazoles: A New Class of Inhibitors with Hypoglycemiant Activity


    Volume 13, Issue 11, July 23, 2012, Pages: 1584–1593, Prof. Dr. Mario Roberto Senger, Lucas da Costa Andrade Gomes, Prof. Dr. Sabrina Baptista Ferreira, Prof. Dr. Carlos Roland Kaiser, Prof. Dr. Vitor Francisco Ferreira and Prof. Dr. Floriano Paes Silva Jr

    Article first published online : 29 JUN 2012, DOI: 10.1002/cbic.201200272

  7. Bicyclic Peptide Inhibitor of Urokinase-Type Plasminogen Activator: Mode of Action


    Volume 14, Issue 16, November 4, 2013, Pages: 2179–2188, Dr. Renée Roodbeen, Berit Paaske, Longguang Jiang, Dr. Jan K. Jensen, Anni Christensen, Dr. Jakob T. Nielsen, Prof. Dr. Mingdong Huang, Prof. Frans A. A. Mulder, Prof. Dr. Niels Chr. Nielsen, Prof. Dr. Peter A. Andreasen and Prof. Dr. Knud J. Jensen

    Article first published online : 2 OCT 2013, DOI: 10.1002/cbic.201300335

  8. Type II Ligands as Chemical Auxiliaries To Favor Enzymatic Transformations by P450 2E1


    Volume 13, Issue 17, November 26, 2012, Pages: 2527–2536, Amélie Ménard, Camilo Fabra, Yue Huang and Prof. Karine Auclair

    Article first published online : 5 NOV 2012, DOI: 10.1002/cbic.201200524

  9. Chemoenzymatic Synthesis of Trehalose Analogues: Rapid Access to Chemical Probes for Investigating Mycobacteria


    Bailey L. Urbanek, Douglas C. Wing, Krystal S. Haislop, Chelsey J. Hamel, Dr. Rainer Kalscheuer, Prof. Peter J. Woodruff and Prof. Benjamin M. Swarts

    Article first published online : 19 AUG 2014, DOI: 10.1002/cbic.201402288

  10. A Conserved Tyrosine in Ferritin Is a Molecular Capacitor


    Volume 14, Issue 9, June 17, 2013, Pages: 1123–1133, Kourosh Honarmand Ebrahimi, Dr. Peter-Leon Hagedoorn and Prof. Dr. Wilfred R. Hagen

    Article first published online : 4 JUN 2013, DOI: 10.1002/cbic.201300149

  11. Significantly Enhanced DNA Thermal Stability Resulting from Porphyrin H-Aggregate Formation in the Minor Groove of the Duplex


    Volume 11, Issue 13, September 3, 2010, Pages: 1833–1839, Adam W. I. Stephenson, Niels Bomholt, Ashton C. Partridge and Vyacheslav V. Filichev

    Article first published online : 30 JUL 2010, DOI: 10.1002/cbic.201000326

  12. Progress and Prospects of Pyrrole-Imidazole Polyamide–Fluorophore Conjugates as Sequence-Selective DNA Probes


    Volume 13, Issue 15, October 15, 2012, Pages: 2170–2185, Dr. Thangavel Vaijayanthi, Dr. Toshikazu Bando, Dr. Ganesh N. Pandian and Prof. Dr. Hiroshi Sugiyama

    Article first published online : 28 SEP 2012, DOI: 10.1002/cbic.201200451

  13. Synthesis of 5,6-Spiroethers and Evaluation of their Affinities for the Bacterial A Site


    Volume 12, Issue 8, May 16, 2011, Pages: 1188–1192, Dr. Ioannis A. Katsoulis, Dr. Georgia Kythreoti, Dr. Athanasios Papakyriakou, Konstantina Koltsida, Panoula Anastasopoulou, Dr. Christos I. Stathakis, Ioannis Mavridis, Dr. Thomas Cottin, Emmanuel Saridakis and Dr. Dionisios Vourloumis

    Article first published online : 6 MAY 2011, DOI: 10.1002/cbic.201100076

  14. Development of Selective Inhibitors for Human Aldehyde Dehydrogenase 3A1 (ALDH3A1) for the Enhancement of Cyclophosphamide Cytotoxicity


    Volume 15, Issue 5, March 21, 2014, Pages: 701–712, Dr. Bibek Parajuli, Prof. Dr. Taxiarchis M. Georgiadis, Prof. Dr. Melissa L. Fishel and Prof. Dr. Thomas D. Hurley

    Article first published online : 13 FEB 2014, DOI: 10.1002/cbic.201300625

  15. α-Crystallin Modulates its Chaperone Activity by Varying the Exposed Surface


    Volume 14, Issue 17, November 25, 2013, Pages: 2362–2370, Dr. Valentina Palmieri, Dr. Giuseppe Maulucci, Dr. Alessando Maiorana, Dr. Massimiliano Papi and Prof. Marco De Spirito

    Article first published online : 12 NOV 2013, DOI: 10.1002/cbic.201300447

  16. Development of Fragment-Based n-FABS NMR Screening Applied to the Membrane Enzyme FAAH


    Volume 14, Issue 13, September 2, 2013, Pages: 1611–1619, Chiara Lambruschini, Marina Veronesi, Dr. Elisa Romeo, Dr. Gianpiero Garau, Dr. Tiziano Bandiera, Prof. Dr. Daniele Piomelli, Dr. Rita Scarpelli and Dr. Claudio Dalvit

    Article first published online : 5 AUG 2013, DOI: 10.1002/cbic.201300347

  17. Recent Developments in the Application of Baeyer–Villiger Monooxygenases as Biocatalysts


    Volume 11, Issue 16, November 2, 2010, Pages: 2208–2231, Dr. Gonzalo de Gonzalo, Prof. Dr. Marko D. Mihovilovic and Prof. Dr. Marco W. Fraaije

    Article first published online : 8 OCT 2010, DOI: 10.1002/cbic.201000395

  18. A Tailor-Made “Tag–Receptor” Affinity Pair for the Purification of Fusion Proteins


    Volume 15, Issue 10, July 7, 2014, Pages: 1423–1435, Dr. Ana S. Pina, Dr. Márcia Guilherme, Prof. Alice S. Pereira, Cláudia S. M. Fernandes, Dr. Ricardo J. F. Branco, Dr. Graziella El Khoury, Prof. Christopher R. Lowe and Prof. A. Cecília A. Roque

    Article first published online : 5 JUN 2014, DOI: 10.1002/cbic.201400018

  19. Design and Synthesis of Selenazole-Containing Peptides for Cocrystallization with P-Glycoprotein


    Volume 12, Issue 6, April 11, 2011, Pages: 868–873, Dr. Houchao Tao, Yue Weng, Dr. Rupeng Zhuo, Prof. Dr. Geoffrey Chang, Prof. Dr. Ina L. Urbatsch and Prof. Dr. Qinghai Zhang

    Article first published online : 8 MAR 2011, DOI: 10.1002/cbic.201100048

  20. Selective Inhibition of an Apicoplastic Aminoacyl-tRNA Synthetase from Plasmodium falciparum


    Volume 14, Issue 4, March 4, 2013, Pages: 499–509, Dr. Rob Hoen, Dr. Eva Maria Novoa, Alba López, Noelia Camacho, Dr. Laia Cubells, Pedro Vieira, Prof. Manuel Santos, Patricia Marin-Garcia, Prof. Jose Maria Bautista, Prof. Alfred Cortés, Prof. Lluís Ribas de Pouplana and Dr. Miriam Royo

    Article first published online : 27 FEB 2013, DOI: 10.1002/cbic.201200620