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There are 2202 results for: content related to: Synthesis and Anti-herpetic Activity of Phosphoramidate ProTides

  1. Prodrugs of butyric acid from bench to bedside: Synthetic design, mechanisms of action, and clinical applications

    Drug Development Research

    Volume 50, Issue 3-4, July - August 2000, Pages: 379–391, Ada Rephaeli, Regina Zhuk and Abraham Nudelman

    Article first published online : 16 OCT 2000, DOI: 10.1002/1098-2299(200007/08)50:3/4<379::AID-DDR20>3.0.CO;2-8

  2. Pivalase Catalytic Antibodies: Towards Abzymatic Activation of Prodrugs

    Chemistry - A European Journal

    Volume 7, Issue 21, November 5, 2001, Pages: 4604–4612, Nicolas Bensel, Martine T. Reymond and Jean-Louis Reymond

    Article first published online : 30 OCT 2001, DOI: 10.1002/1521-3765(20011105)7:21<4604::AID-CHEM4604>3.0.CO;2-Z


    Enzyme Technologies: Pluripotent Players in Discovering Therapeutic Agents

    Ivan S. Krylov, Charles E. McKenna, Pages: 253–300, 2013

    Published Online : 6 DEC 2013, DOI: 10.1002/9781118739907.ch7

  4. γ-Substituted Bis(pivaloyloxymethyl)ester Analogues of Fosmidomycin and FR900098

    Archiv der Pharmazie

    Volume 340, Issue 12, December 2007, Pages: 661–666, Thomas Kurz, Christoph Behrendt, Miriam Pein, Uwe Kaula, Bärbel Bergmann and Rolf D. Walter

    Article first published online : 12 NOV 2007, DOI: 10.1002/ardp.200700107

  5. Prodrugs of 6-thiopurines: Enhanced delivery through the skin

    Journal of Pharmaceutical Sciences

    Volume 72, Issue 4, April 1983, Pages: 372–378, K. B. Sloan, M. Hashida, J. Alexander, N. Bodor and T. Higuchi

    Article first published online : 22 SEP 2006, DOI: 10.1002/jps.2600720413

  6. In vitro, ex vivo, and in situ intestinal absorption characteristics of the antiviral ester prodrug adefovir dipivoxil

    Journal of Pharmaceutical Sciences

    Volume 89, Issue 8, August 2000, Pages: 1054–1062, Pieter Annaert, Josef J. Tukker, Jan van Gelder, Lieve Naesens, Erik de Clercq, Guy van den Mooter, Renaat Kinget and Patrick Augustijns

    Article first published online : 18 JUL 2000, DOI: 10.1002/1520-6017(200008)89:8<1054::AID-JPS10>3.0.CO;2-5

  7. Rearrangement process occurring in the fragmentation of adefovir derivatives

    Journal of Mass Spectrometry

    Volume 39, Issue 2, February 2004, Pages: 145–152, Xiaoyan Chen, Jie Xing and Dafang Zhong

    Article first published online : 18 FEB 2004, DOI: 10.1002/jms.557

  8. You have full text access to this OnlineOpen article
    In vivo and in vitro antitumor activity of butyroyloxymethyl-diethyl phosphate (AN-7), a histone deacetylase inhibitor, in human prostate cancer

    International Journal of Cancer

    Volume 116, Issue 2, 20 August 2005, Pages: 226–235, Ada Rephaeli, Diana Blank-Porat, Nataly Tarasenko, Michal Entin-Meer, Inesa Levovich, Suzanne M. Cutts, Don R. Phillips, Zvi Malik and Abraham Nudelman

    Article first published online : 30 MAR 2005, DOI: 10.1002/ijc.21030

  9. Effects of vehicles and prodrug properties and their interactions on the delivery of 6-mercaptopurine through skin: S6-acyloxymethyl-6-mercaptopurine prodrugs

    Journal of Pharmaceutical Sciences

    Volume 77, Issue 3, March 1988, Pages: 210–215, Robert P. Waranis and Kenneth B. Sloan

    Article first published online : 21 SEP 2006, DOI: 10.1002/jps.2600770306

  10. [2+2] Photocycloaddition of Symmetrically Disubstituted Alkenes to 2(5H)-Furanones: Diastereoselective Entry to 1,2,3,4-Tetrasubstituted Cyclobutanes

    European Journal of Organic Chemistry

    Volume 2011, Issue 20-21, July 2011, Pages: 3888–3895, Sònia Parés, Pedro de March, Josep Font, Ramon Alibés and Marta Figueredo

    Article first published online : 6 MAY 2011, DOI: 10.1002/ejoc.201100067

  11. Chemical Synthesis of RNA with Base-Labile 2′-O-(Pivaloyloxymethyl)-Protected Ribonucleoside Phosphoramidites


    Current Protocols in Nucleic Acid Chemistry


    Thomas Lavergne, Michaël Janin, Christelle Dupouy, Jean-Jacques Vasseur and Françoise Debart

    Published Online : 1 DEC 2010, DOI: 10.1002/0471142700.nc0319s43

  12. Structure of pivaloyloxymethyl (3S,5R)-6,6-dibromopenicillanate 1,1-dioxide

    Acta Crystallographica Section C

    Volume 42, Issue 8, August 1986, Pages: 1029–1032, P. M. Alzari, B. E. Rivero, G. Punte and A. E. Ronco

    DOI: 10.1107/S0108270186093605

  13. Synthesis of Oligodeoxynucleotides Containing 5-(β-D-Glucopyranosyloxymethyl)-2′-deoxyuridine, a Modified Nucleoside in the DNA of Trypanosoma Brucei

    European Journal of Organic Chemistry

    Volume 1999, Issue 9, September 1999, Pages: 2337–2344, Martin de Kort, Edwin Ebrahimi, Eric R. Wijsman, Gijs A. van der Marel and Jacques H. van Boom

    Article first published online : 12 AUG 1999, DOI: 10.1002/(SICI)1099-0690(199909)1999:9<2337::AID-EJOC2337>3.0.CO;2-F

  14. Effect of aminomethyl (N-mannich base) derivatization on the ability of S6-acetyloxymethyl-6-mercaptopurine prodrug to deliver 6-mercaptopurine through hairless mouse skin

    Journal of Pharmaceutical Sciences

    Volume 79, Issue 12, December 1990, Pages: 1099–1104, Akram N. Saab, Kenneth B. Sloan, Howard D. Beall and René Villanueva

    Article first published online : 17 SEP 2006, DOI: 10.1002/jps.2600791212

  15. Pivaloxymethyl chloride

    Standard Article

    e-EROS Encyclopedia of Reagents for Organic Synthesis

    Jean-Paul Desaulniers

    Published Online : 15 MAR 2011, DOI: 10.1002/047084289X.rn01252

  16. 1-Alkylcarbonyloxymethyl prodrugs of 5-fluorouracil (5-FU): Synthesis, physicochemical properties, and topical delivery of 5-FU

    Journal of Pharmaceutical Sciences

    Volume 87, Issue 1, January 1998, Pages: 15–20, H. Elizabeth Taylor and Kenneth B. Sloan

    Article first published online : 12 JUN 2000, DOI: 10.1021/js9702574

  17. ChemInform Abstract: Stereoselective Reduction of Pivaloyloxymethyl (2S,5R,6S)-6-Acetyl-3,3- dimethyl-7-oxo-4-thia-1-azabicyclo(3.2.0)heptane-2-carboxylate with Sodium Borohydride.


    Volume 23, Issue 36, September 8, 1992, Page: no, D. DONATI, C. MARCHIORO, B. TAMBURINI and A. URSINI

    Article first published online : 21 AUG 2010, DOI: 10.1002/chin.199236275

  18. Pharmacokinetics of Pradefovir and PMEA in Healthy Volunteers After Oral Dosing of Pradefovir

    The Journal of Clinical Pharmacology

    Volume 45, Issue 11, November 2005, Pages: 1250–1258, Chin-chung Lin, Christine Xu, Alice Teng, Li-Tain Yeh and Janet Peterson

    Article first published online : 8 MAR 2013, DOI: 10.1177/0091270005280644

  19. Easy preparative scale syntheses of labelled xanthines: caffeine, theophylline and theobromine

    Journal of Labelled Compounds and Radiopharmaceuticals

    Volume 50, Issue 1, 2007, Pages: 33–41, Frédéric Balssa and Yves Bonnaire

    Article first published online : 22 JAN 2007, DOI: 10.1002/jlcr.1154

  20. REVIEW: Present and future directions in the treatment of chronic hepatitis B infection

    Journal of Gastroenterology and Hepatology

    Volume 12, Issue 12, December 1997, Pages: 843–854, AMANDA NICOLL and STEPHEN LOCARNINI

    Article first published online : 28 JUN 2008, DOI: 10.1111/j.1440-1746.1997.tb00382.x