Chapter 16. Synthesis of Enantiopure Azasugars from D-Mannitol: Carbohydrate and Peptide Mimics
- Yves Chapleur
Published Online: 28 JAN 2005
DOI: 10.1002/3527603239.ch16
Copyright © 1998 Wiley-VCH Verlag GmbH
Book Title
Carbohydrate Mimics: Concepts and Methods
Additional Information
How to Cite
Depezay, J.-C. (2005) Synthesis of Enantiopure Azasugars from D-Mannitol: Carbohydrate and Peptide Mimics, in Carbohydrate Mimics: Concepts and Methods (ed Y. Chapleur), Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim, FRG. doi: 10.1002/3527603239.ch16
Editor Information
UMR CNRS 7565, Université Henri Poincaré-Nancy I, BP239, F-54506 Vandceuvre, France
Publication History
- Published Online: 28 JAN 2005
- Published Print: 12 NOV 1997
ISBN Information
Print ISBN: 9783527295265
Online ISBN: 9783527603237
- Summary
- Chapter
Keywords:
- enantiopure;
- azasugars;
- D-mannitol;
- carbohydrate;
- peptide;
- bis-aziridines;
- azadisaccharides;
- bis-epoxides;
- somatostatin
Summary
Introduction
Results
To Azasugars via Bis-Aziridines
Nucleophilic Opening of Bis-Aziridines
Bis-Aziridines Precursors of Azadisaccharides
To Azasugars via Bis-Epoxides
Nucleophilic Opening of Bis-Epoxides
Isomerisation of Polyhydroxylated Piperidines
Isomerisation of Polyhydroxylated Azepanes
Inhibition Studies
Synthesis of Non-Peptide Mimics of Somatostatin
Conclusion
References