Chapter 19. Protein Kinase Structural Biology: Methods and Strategies for Targeted Drug Discovery
- Rongshi Li,
- Jeffrey A. Stafford
Published Online: 28 SEP 2009
DOI: 10.1002/9780470524961.ch19
Copyright © 2009 John Wiley & Sons, Inc.
Book Title
Kinase Inhibitor Drugs
Additional Information
How to Cite
Mol, C. D., Okada, K. and Hosfield, D. J. (2009) Protein Kinase Structural Biology: Methods and Strategies for Targeted Drug Discovery, in Kinase Inhibitor Drugs (eds R. Li and J. A. Stafford), John Wiley & Sons, Inc., Hoboken, NJ, USA. doi: 10.1002/9780470524961.ch19
Editor Information
Takeda San Diego, Inc., San Diego, CA 92121, USA
Publication History
- Published Online: 28 SEP 2009
- Published Print: 2 OCT 2009
ISBN Information
Print ISBN: 9780470278291
Online ISBN: 9780470524961
- Summary
- Chapter
- References
Keywords:
- protein kinase structural biology - targeted drug discovery strategies;
- kinase inhibition and targeting allosteric sites;
- kinase inhibition by targeting active conformations
Summary
This chapter contains sections titled:
Introduction
Methods for Kinase Structural Biology
Kinase Architecture
Kinase Inhibition by Targeting Active Conformations
Kinase Inhibition by Targeting Inactive Conformations
Kinase Inhibition by Targeting Allosteric Sites
Summary and Perspectives
References