18. Azaindole Hydroxamic Acids are HIV-1 Integrase Inhibitors
- Nouri Neamati
Published Online: 28 SEP 2011
DOI: 10.1002/9781118015377.ch18
Copyright © 2011 John Wiley & Sons, Inc.
Book Title
HIV-1 Integrase: Mechanism and Inhibitor Design
Additional Information
How to Cite
Plewe, M. B. and Johnson, T. W. (2011) Azaindole Hydroxamic Acids are HIV-1 Integrase Inhibitors, in HIV-1 Integrase: Mechanism and Inhibitor Design (ed N. Neamati), John Wiley & Sons, Inc., Hoboken, NJ, USA. doi: 10.1002/9781118015377.ch18
Editor Information
Department of Pharmacology and Pharmaceutical Sciences, University of Southern California, School of Pharmacy, Los Angeles, California, USA
Publication History
- Published Online: 28 SEP 2011
- Published Print: 9 SEP 2011
ISBN Information
Print ISBN: 9780470184745
Online ISBN: 9781118015377
- Summary
- Chapter
- References
Keywords:
- azaindole hydroxamic acids, HIV-1 inhibitors;
- high-throughput screening;
- azaindole hydroxamic acid mutagenicity
Summary
This chapter contains sections titled:
Introduction
High-Throughput Screening
Azaindole Hydroxamic Acids
β-Carboline Hydroxamic Acids
Picoline Hydroxamic Acids
Mutagenicity of Azaindole Hydroxamic Acids
Metabolic Stability of Azaindole Hydroxamic Acids
Synthesis
Conclusions
Acknowledgments
References