Palladium-Catalyzed Amination of Aryl Mesylates

Authors

  • Chau Ming So,

    1. Open Laboratory of Chirotechnology of the Institute of Molecular Technology for Drug Discovery and Synthesis and Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong (Hong Kong), Fax: (+852) 2364-9932
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  • Zhongyuan Zhou Prof. Dr.,

    1. Open Laboratory of Chirotechnology of the Institute of Molecular Technology for Drug Discovery and Synthesis and Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong (Hong Kong), Fax: (+852) 2364-9932
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  • Chak Po Lau Prof. Dr.,

    1. Open Laboratory of Chirotechnology of the Institute of Molecular Technology for Drug Discovery and Synthesis and Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong (Hong Kong), Fax: (+852) 2364-9932
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  • Fuk Yee Kwong Prof. Dr.

    1. Open Laboratory of Chirotechnology of the Institute of Molecular Technology for Drug Discovery and Synthesis and Department of Applied Biology and Chemical Technology, The Hong Kong Polytechnic University, Hung Hom, Kowloon, Hong Kong (Hong Kong), Fax: (+852) 2364-9932
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  • We thank the Research Grants Council of Hong Kong (Project No. CERG: PolyU5008/06P) and University Grants Committee Areas of Excellence Scheme (Project No. AoE/P-10/01) for financial support.

Abstract

original image

Kein Problem mit Wasser: Der Phosphanligand L und Pd(OAc)2 als Vorstufe ermöglichen die erste palladiumkatalysierte Aminierung nichtaktivierter Arylmesylate. Das Katalysatorsystem kann in einem wässrigen Reaktionsmedium ohne nachteilige Effekte eingesetzt werden.

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