Sulfonyl-1,2,3-Triazoles: Convenient Synthones for Heterocyclic Compounds

Authors


  • This work was supported by the National Science Foundation (CHE-0848982)

Abstract

original image

As easy as 1,2,3: Readily available and shelf-stable 1-sulfonyl-1,2,3-triazoles react with aldehydes and aldimines in the presence of RhII catalysts to produce 4-oxazolines and 1,2,5-trisubstituted imidazoles (see scheme).

Ancillary