Financial support for this work was provided by the NIH/NIGMS (GM-073949), Eisai, the Binational US-Israel Science Foundation, and the Frost Foundation (to D.S). We are grateful to P. Siva (Bristol-Myers Squibb) for the calculations shown in Scheme 1 A, to J. Kadow (Bristol-Myers Squibb) for a sample of 36, and to T. Ryba and C. Thomas (Sigma–Aldrich) for a donation of chemicals. The Uehara Memorial Foundation and SIOC provided funding for postdoctoral fellowships to Y.F. and Q.Z., respectively.
Direct Synthesis of Fluorinated Heteroarylether Bioisosteres†
Article first published online: 4 MAR 2013
Copyright © 2013 WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim
Angewandte Chemie International Edition
Volume 52, Issue 14, pages 3949–3952, April 2, 2013
How to Cite
Zhou, Q., Ruffoni, A., Gianatassio, R., Fujiwara, Y., Sella, E., Shabat, D. and Baran, P. S. (2013), Direct Synthesis of Fluorinated Heteroarylether Bioisosteres . Angew. Chem. Int. Ed., 52: 3949–3952. doi: 10.1002/anie.201300763
- Issue published online: 26 MAR 2013
- Article first published online: 4 MAR 2013
- Manuscript Received: 29 JAN 2013
- NIH/NIGMS. Grant Number: GM-073949
- Binational US-Israel Science Foundation
- Frost Foundation
- Bristol-Myers Squibb
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