This work was supported by the EPSRC.
2-Aminobenzaldehydes as Versatile Substrates for Rhodium-Catalyzed Alkyne Hydroacylation: Application to Dihydroquinolone Synthesis†
Version of Record online: 12 NOV 2013
© 2013 The Authors. Published by Wiley-VCH Verlag GmbH & Co. KGaA. This is an open access article under the terms of the Creative Commons Attribution License, which permits use, distribution and reproduction in any medium, provided the original work is properly cited.
Angewandte Chemie International Edition
Volume 52, Issue 50, pages 13280–13283, December 9, 2013
How to Cite
Castaing, M., Wason, S. L., Estepa, B., Hooper, J. F. and Willis, M. C. (2013), 2-Aminobenzaldehydes as Versatile Substrates for Rhodium-Catalyzed Alkyne Hydroacylation: Application to Dihydroquinolone Synthesis. Angew. Chem. Int. Ed., 52: 13280–13283. doi: 10.1002/anie.201308127
- Issue online: 5 DEC 2013
- Version of Record online: 12 NOV 2013
- Manuscript Received: 16 SEP 2013
- Funded Access
- 2For reviews, see:
- 3For recent examples, see:
- 4For examples, see:
- 5For examples, see:
- 6For examples, see:
- 8For examples, see:
- 10For examples, see:
- 15See Ref. [4a].
- 27Hydroacylation adducts derived from primary amines could be directly converted into dihydroquinolones without purification, provided that a solvent swap (acetone to MeCN) was performed before addition of SbCl3.