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Keywords:

  • Aurora A;
  • fluorescent probes;
  • inhibitors;
  • kinetics;
  • protein kinases;
  • residence time
Thumbnail image of graphical abstract

The inside cover picture shows fluorescent probes based on well-known inhibitors MLN8237 and VX-689 (MK-5108) that revealed slow association/dissociation kinetics in inhibition and binding assays with Aurora A kinase. For more details see the paper by D. Lavõgina et al. on p. 443 ff.