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A General and Efficient Palladium-Catalyzed Carbonylative Synthesis of 2-Aryloxazolines and 2-Aryloxazines from Aryl Bromides

Authors

  • Dr. Xiao-Feng Wu,

    Corresponding author
    1. Department of Chemistry, Zhejiang Sci-Tech University, Xiasha Campus, Hangzhou, Zhejiang Province, 310018 (P.R. China)
    2. Leibniz-Institut für Katalyse e.V. an der Universitüt Rostock, Albert-Einstein-Strasse 29a, 18059 Rostock (Germany), Fax: (+49) 381-1281-5000
    • Department of Chemistry, Zhejiang Sci-Tech University, Xiasha Campus, Hangzhou, Zhejiang Province, 310018 (P.R. China)
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  • Dr. Helfried Neumann,

    1. Leibniz-Institut für Katalyse e.V. an der Universitüt Rostock, Albert-Einstein-Strasse 29a, 18059 Rostock (Germany), Fax: (+49) 381-1281-5000
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  • Stephan Neumann,

    1. Leibniz-Institut für Katalyse e.V. an der Universitüt Rostock, Albert-Einstein-Strasse 29a, 18059 Rostock (Germany), Fax: (+49) 381-1281-5000
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  • Prof. Dr. Matthias Beller

    Corresponding author
    1. Leibniz-Institut für Katalyse e.V. an der Universitüt Rostock, Albert-Einstein-Strasse 29a, 18059 Rostock (Germany), Fax: (+49) 381-1281-5000
    • Leibniz-Institut für Katalyse e.V. an der Universitüt Rostock, Albert-Einstein-Strasse 29a, 18059 Rostock (Germany), Fax: (+49) 381-1281-5000
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Abstract

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Oxazoline is OK! A general and efficient method for the synthesis of oxazolines has been developed (see scheme). This allowed the preparation of 27 five-membered-ring heterocycles and 11 six-membered-ring heterocycles in moderate to good yields.

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