Iron(III)-Catalyzed Direct N-Alkylation of Azoles via Oxidative Transformation of sp3 C[BOND]H Bonds under Solvent-Free Conditions

Authors

  • Xiang Liu,

    1. State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China
    2. Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Lanzhou, Gansu 730000, China
    Search for more papers by this author
  • Yongxin Chen,

    1. State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China
    2. Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Lanzhou, Gansu 730000, China
    Search for more papers by this author
  • Kangning Li,

    1. State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China
    2. Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Lanzhou, Gansu 730000, China
    Search for more papers by this author
  • Dong Wang,

    1. State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China
    2. Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Lanzhou, Gansu 730000, China
    Search for more papers by this author
  • Baohua Chen

    Corresponding author
    1. State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China
    2. Key Laboratory of Nonferrous Metal Chemistry and Resources Utilization of Gansu Province, Lanzhou, Gansu 730000, China
    • State Key Laboratory of Applied Organic Chemistry, Lanzhou University, Lanzhou, Gansu 730000, China, Tel.: 0086-0139-193-57881; Fax: 0086-0931-891-2582
    Search for more papers by this author

Abstract

A new approach to synthesize N-alkylation of azoles by iron(III)-catalyst under solvent-free conditions was developed. The method is broad in scope and highly efficient.

Ancillary