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Keywords:

  • acylguanidines;
  • bioisosterism;
  • neuropeptide Y;
  • radiochemistry;
  • radioligands
Thumbnail image of graphical abstract

Radioing in on NPY: Attachment of a [2,3-3H]propionyl group through an appropriate linker to the guanidine group of an (S)-argininamide-type neuropeptide Y (NPY) Y2 receptor antagonist resulted in a subtype-selective radioligand.