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  • BIRCH, P.J., HAYES, A.G. & SHEEHAN, M.J. (1987). Intrathecal administration of δ-selective opioid peptides produces antinociception mediated via μ-receptors. Abstracts Br. Opioid Coll., P2, Oxford.
  • CHENG, Y.C. & PRUSOFF, W.H. (1973). Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymic reaction. Biochem. Pharmacol., 22, 30993108.
  • CLARK, C.R., MORE, B. BIRCH, SHARIF, N.A., HUNTER, J.C., HILL, R.G. & HUGHES, J. (1988). PD 117302: a selective agonist for the κ-opioid receptor. Br. J. Pharmacol., 93, 618626.
  • COTTON, R., GILES, M.G., MILLER, L., SHAW, J.S. & TIMMS, D. (1984). ICI 174864. A highly selective antagonist at the opioid delta receptor. Eur. J. Pharmacol., 97, 331332.
  • COTTON, R., KOSTERLITZ, H.W., PATERSON, S.J., RANCE, M.J. & TRAYNOR, J.R. (1985). The use of [3H]-[d-Pen2,d-Pen5]enkephalin as a highly selective ligand for the δ-binding site. Br. J. Pharmacol., 84, 927932.
  • COWAN, A., RANCE, M.J. & BLACKBURN, T.P. (1986). In vivo studies on delta opioid receptors. In NIDA Research Monograph 75, Progress in Opioid Research, ed. Holaday, J.W., Law, P.-Y. & Herz, A. pp. 473476. Maryland, U.S.A.: National Institute of Drug Abuse.
  • CZLONKOWSKI, A., COSTA, T., PRZWLOCKI, R., PASI, A. & HERZ, A. (1983). Opiate receptor binding sites in human spinal cord. Brain Res., 267, 392396.
  • DELEAN, A., MUNSON, P.J. & RODBARD, D. (1978). Simultaneous analysis of families of sigmoid curves: application to bioassay, radioligand assay, and physiological dose-response curves. Am. J. Physiol., 235, E97102.
  • GORMLEY, J.J., MORLEY, J.S., PRIESTLEY, T., SHAW, J.S., TURNBULL, M.J. & WHEELER, H. (1982). In vivo evaluation of the opiate delta receptor antagonist ICI 154,129. Life Sci., 31, 12631266.
  • GOUARDERES, C., ATTALI, B., AUDIGIER, Y. & CROS, J. (1983). Interaction of selective mu and delta ligands with the kappa2 subtype of opiate binding sites. Life Sci., 33 (suppl. 1), 175178.
  • HEYMAN, J.S., KOSLO, R.J., MOSBERG, H.J., TALLARIDA, R.J. & PORRECA, F. (1986). Estimation of the affinity of naloxone at supraspinal and spinal opioid receptors in vivo: studies with receptor selective agonists. Life Sci., 39, 17951803.
  • HEYMAN, J.S., MULVANEY, S.A., MOSBERG, H.I. & PORRECA, F. (1987). Opioid δ-receptor involvement in supraspinal and spinal antinociception in mice. Brain Res., 420, 100108.
  • HILL, A.W. (1910). The possible effects of the aggregation of the molecules of haemoglobin on its dissociation curves. J. Physiol., 40, iv-vii.
  • HYLDEN, J.L.K. & WILCOX, G.L. (1980). Intrathecal morphine in mice: a new technique. Eur. J. Pharmacol., 67, 313316.
  • LEIGHTON, G.E., RODRIGUEZ, R.E., HILL, R.G. & HUGHES, J. (1988). κ-opioid agonists produce antinociception after i.v. and i.c.v., but not intrathecal administration in the rat. Br. J. Pharmacol., 93, 553560.
  • LESLIE, F. M. (1987). Methods used for the study of opioid receptors. Pharmacol. Rev., 39, 197249.
  • MARTIN, W.R., EADES, C.G. THOMPSON, J.A., HUPPLER, R.E. & GILBERT, P.E. (1976). The effects of morphine and nalorphine-like drugs in the non-dependent and morphine dependent chronic spinal dog. J. Pharmacol. Exp. Ther., 197, 517532.
  • McPHERSON, G.A. (1985). Analysis of radioligand binding experiments. J. Pharmacol. Meth., 14, 213228.
  • MEUNIER, J.-C., KOUAKOU, Y., PUGET, A. & MOISAND, C. (1983). Multiple opiate binding sites in the central nervous system of the rabbit. Mol. Pharmacol., 24, 2329.
  • MOSBERG, H.I., HURST, R., HRUBY, V.J., GEE, K., YAMAMURA, H.J., GALLIGAN, J.E. & BURKS, T.F. (1983). Bis-penicillamine enkephalins possess highly improved specificity towards δ-opioid receptors. Proc. Natl. Acad. Sci. U.S.A., 80, 58715874.
  • PORRECA, F., HEYMAN, J.S., MOSBERG, H.J., OMNAS, J.R. & VAUGHT, J.L. (1987a). Role of mu and delta receptors in the supraspinal and spinal analgesic effects of [d-Pen2,d-Pen5]enkephalin in the mouse. J. Pharmacol. Exp. Ther., 241, 393399.
  • PORRECA, F., MOSBERG, H.I., HURST, R., HRUBY, V.J. & BURKS, T.F. (1984). Roles of mu, delta and kappa opioid receptors in spinal and supraspinal mediation of gastrointestinal transit effects and hot-plate analgesia in the mouse. J. Pharmacol. Exp. Ther., 230, 341348.
  • PORRECA, F., MOSBERG, H.I., OMNAS, J.R., BURKS, T.F. & COWAN, A. (1987b). Supraspinal and spinal potency of selective opioid agonists in the mouse writhing test. J. Pharmacol. Exp. Ther., 240, 890894.
  • ROBSON, L.E., GILLAN, M.C.G. & KOSTERLITZ, H.W. (1985). Species differences in the concentrations and distributions of opioid binding sites. Eur. J. Pharmacol., 112, 6571.
  • ROTHMAN, R.B., DANKS, J.A., JACOBSON, A.E., BURKE, T.R. & RICE, K.C. (1985). Leucine enkephalin noncompetitively inhibits the binding of [3H]naloxone to the opiate mu-recognition site: evidence for delta-mu binding site interactions in vitro. Neuropeptides, 6, 351363.
  • RODRIGUEZ, R.E., LEIGHTON, G., HILL, R.G. & HUGHES, J. (1986). In vivo evidence for spinal delta-opiate receptor-operated antinociception. Neuropeptides, 8, 221241.
  • SCATCHARD, G. (1949). The attractions of proteins for small molecules and ions. Ann. New York Acad. Sci., 51, 660672.
  • SCHMAUSS, C. & YAKSH, T.L. (1984). In vivo studies on spinal opiate receptor systems mediating antinociception. II Pharmacological profiles suggesting a differential association of mu, delta and kappa receptors with visceral chemical and cutaneous thermal stimuli in the rat. J. Pharmacol. Exp. Ther., 228, 112.
  • TRAYNOR, J.R., HILL, R.G., HUGHES, J., HUNTER, J.C. & RODRIGUEZ, R.E. (1988). Delta opioid binding sites in the spinal cords of various rodents. Br. J. Pharmacol., 94, 375P.
  • TRAYNOR, J.R. & RANCE, M.J. (1984). Opiate binding in the rat spinal cord: evidence for mu and delta sites. Neuropeptides, 5, 8184.
  • TRAYNOR, J.R. & WOOD, M.S. (1987). Distribution of opioid binding sites in spinal cord. Neuropeptides, 10, 313320.
  • TUNG, A.S. & YAKSH, T.L. (1982). In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord. Brain Res., 247, 7583.
  • YAKSH, T.L. (1983). In vivo studies on spinal opiate receptors mediating antinociception. I. mu and delta receptor profiles in the primate. J. Pharmacol. Exp. Ther., 226, 303316.
  • YAKSH, T.L. & NOUEIHED, R.L. (1985). The physiology and pharmacology of spinal opiates. Ann. Rev. Pharmacol. Toxicol., 25, 433462.
  • ZARR, C.D., WERLING, L.L., BROWN, S.R. & COX, B.M. (1986). Opioid ligand binding sites in the spinal cord of the guinea-pig. Neuropharmacology, 25, 471480.