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References

  • CHEUNG, H.S., WANG, F.L., ONDETTI, M.A., SABO, E.F. & CUSHMAN, D.W. (1980). Binding of peptide substrates and inhibitors of angiotensin-converting enzyme. J. Biol. Chem., 255, 401407.
  • DANTZIG, A.H. & BERGIN, L. (1990). Uptake of the cephalosporin, cephalexin, by a dipeptide transport carrier in the human intestinal cell line, Caco-2. Biochim. Biophys. Acta, 1027, 211217.
  • DUCHIN, K.L., SINGHVI, S.M., WILLARD, D.A., MIGDALOF, B.H. & McKINSTRY, D.N. (1982). Captopril kinetics. Clin. Pharmacol. Then, 31, 452457.
  • FEI, Y.J., KANAI, Y., NUSSBERGER, S., GANAPATHY, V., LEIBACH, F.H., ROMERO, M.F., SINGH, S.K., BORON, W.F. & HEDIGER, M.W. (1994). Expression cloning of a mammalian proton-coupled oligopeptide transporter. Nature, 368, 563566.
  • FRIEDMAN, D.I. & AMIDON, G.L. (1989a). Passive and carrier-mediated intestinal absorption components of two angiotensin converting enzyme (ACE) inhibitor prodrugs in rats: enalapril and fosinopril. Pharmacol. Res., 6, 10431047.
  • FRIEDMAN, D.I. & AMIDON, G.L. (1989b). Intestinal absorption mechanisms of dipeptide angiotensin converting enzyme inhibitors of the lysyl-proline type: lisinopril and SQ 29,852, J. Pharmacol. Sci., 78, 995998.
  • GANAPATHY, V. & LEIBACH, F.H. (1985). Is intestinal peptide transport energized by a proton gradient Am. J. Physiol., 249, G153G160.
  • HIDALGO, I.J., RAUB, T.J. & BORCHARDT, R.T. (1989). Characterisation of the human colonic carcinoma cell line (Caco-2) as a model system for intestinal epithelial permeability. Gastroenterology, 96, 736749.
  • HU, M. & AMIDON, G.L. (1988). Passive and carrier-mediated intestinal absorption components of captopril. J. Pharmacol. Sci., 77, 10071011.
  • HUMPHREY, M.J. (1986). The oral bioavailability of peptides and related drugs. In Delivery Systems for Peptide Drugs, ed. Davis, S.S., Hum, L. & Tomlinson, E. pp. 139151. NATO ASI Series 125, New York: Plenum.
  • HUMPHREY, M.L. & RINGROSE, P.S. (1986). Peptides and related drugs: a review of their absorption, metabolism, and excretion. Drug Metab. Rev., 17, 283310.
  • INUI, K.I., YAMAMOTO, M. & SAITO, H. (1992). Transepithelial transport of oral cephalisporins by monolayers of intestinal epithelial cell line Caco-2: specific transport systems in apical and basolateral membranes. J. Pharmacol. Exp. Ther., 261, 195201.
  • LUCAS, M.L., SCHNEIDER, W., HABERICH, F.J. & BLAIR, J.A. (1975). Direct measurement by pH-microelectrode of the pH-microclimate in rat proximal jejunum. Proc. R. Soc. B, 192, 3948.
  • MATTHEWS, D.M. (1975). Absorption of peptides by mammalian intestine. In Peptide Transport in Protein Nutrition. ed. Matthews, D.M. & Payne, J.W., North-Holland research monographs, Frontiers of Biology, 37 pp. 61146. Amsterdam: North Holland.
  • MATTHEWS, D.M. & ADIBI, S.A. (1976). Peptide absorption. Gastroenterology, 71, 151161.
  • McEWAN, G.T.A., DANIEL, H., FETT, C., BURGESS, M.N. & LUCAS, M.L. (1988). The effect of Escherichia coli STa enterotoxin and other secretagogues on mucosal surface pH of rat small intestine in vivo Proc. R. Soc. B, 234, 219237.
  • SAITO, H. & INUI, K.I. (1993). Dipeptide transporters in apical and basolateral membranes of the human intestinal cell line Caco-2. Am. J. Physiol., 265, G289G294.
  • THOMAS, J.A., BUSHBAUM, R.N., ZIMNIAK, A. & RACKER, E. (1979). Intracellular pH measurements in Ehrlich ascites tumour cells utilizing spectroscopic probes generated Biochemistry, 18, 22302238.
  • THWAITES, D.T., BROWN, C.D.A., HIRST, B.H. & SIMMONS, N.L. (1993a). Transepithelial glycylsarcosine transport in intestinal Caco-2 cells mediated by expression of H+-coupled carriers at both apical and basal membranes. J. Biol. Chem., 268, 76407642.
  • THWAITES, D.T., BROWN, C.D.A., HIRST, B.H. & SIMMONS, N.L. (1993b). H+-coupled dipeptide (glycylsarcosine) transport across apical and basal borders of human intestinal Caco-2 cell monolayers display distinctive characteristics. Biochim. Biophys. Acta, 1151, 237245.
  • THWAITES, D.T., HIRST, B.H. & SIMMONS, N.L. (1994a). Substrate specificity of the di/tripeptide transporter in human intestinal epithelia (Caco-2): identification of substrates that undergo H+-coupled absorption. Br. J. Pharmacol., 113, 10501056.
  • THWAITES, D.T., McEWAN, G.T.A., BROWN, C.D.A., HIRST, B.H. & SIMMONS, N.L. (1994b). L-Alanine absorption in human intestinal Caco-2 cells driven by the proton electrochemical gradient. J. Membr. Biol., 140, 143151.
  • THWAITES, D.T., McEWAN, G.T.A., COOK, M.J., HIRST, B.H. & SIMMONS, N.L. (1993c). H+-coupled (Na+-independent) proline transport in human intestinal (Caco-2) epithelial cell monolayers. FEBS Lett., 333, 7882.
  • THWAITES, D.T., McEWAN, G.T.A., HIRST, B.H. & SIMMONS, N.L. (1993d). Transepithelial dipeptide (glycylsarcosine) transport across epithelial monolayers of human Caco-2 cells is rheogenic. Pflügers Arch., 425, 178180.
  • TOCCO, D.J., de LUNA, F.A., DUNCAN, A.E.W., VASSIL, T.C. & ULM, E.H. (1982). The physiological disposition and metabolism of enalapril maleate in laboratory animals. Drug Metab. Disposition, 10, 1519.
  • ULM, E.H., HICHENS, M., GOMEZ, H.J., TILL, A.E., HAND, E., VASSIL, T.C., BIOLLAZ, J., BRUNNER, H.R. & SCHELLING, J.L. (1982). Enalapril maleate and a lysine analogue (MK-521): disposition in man. Br. J. Clin. Pharmacol., 14, 357362.
  • WATSON, A.J.M., LEVINE, S., DONOWITZ, M. & MONTROSE, M.H. (1991). Kinetics and regulation of a polarized Na+-H+ exchanger from Caco-2 cells, a human intestinal cell line. Am. J. Physiol., 261, G229G238.
  • WYVRATT, M.J & PATCHETT, A.A. (1985). Recent developments in the design of angiotensin-converting inhibitors. Med. Res. Rev., 5, 483581.