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Dr. Jing Li, Dr. Tamer S. Kaoud, Jake LeVieux, Brad Gilbreath, Dr. Swapna Moharana, Prof. Kevin N. Dalby and Prof. Sean M. Kerwin A Fluorescence-Based Assay for p38α Recruitment Site Binders: Identification of Rooperol as a Novel p38α Kinase Inhibitor ChemBioChem 14

Version of Record online: 6 DEC 2012 | DOI: 10.1002/cbic.201200529

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A new p38α inhibitor: Using a D-recruitment site (DRS) probe for p38α which exploits covalent interaction with Cys119 and alkyne–azide “click” chemistry to identify small molecules that recognize the p38α DRS, the anti-inflammatory natural product rooperol was identified as a novel p38α inhibitor.

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