European Journal of Organic Chemistry

Cover image for Vol. 2014 Issue 12

Editor: Haymo Ross, Deputy Editor: Susan Wilkinson

Impact Factor: 3.344

ISI Journal Citation Reports © Ranking: 2012: 14/57 (Chemistry Organic)

Online ISSN: 1099-0690

Associated Title(s): Advanced Synthesis & Catalysis, Asian Journal of Organic Chemistry

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Here's a selection of upcoming papers. Also see the EarlyView page for the latest papers published online.

Total Synthesis of (2RS)-α-Tocopherol through Ni-Catalyzed 1,4-Addition to a Chromenone Intermediate
[Short Communications]

Andreas Ole Termath, Janna Velder, René T. Stemmler, Thomas Netscher, Werner Bonrath, Hans-Günther Schmalz*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402240

Enantiospecific Synthesis and Biological Investigations of a Nuphar Alkaloid: Proposed Structure of a Castoreum Component
[Full Papers]

Hajime Seki, Gunda I. Georg*

Coming soon.

First Palladium-Catalyzed Direct Regioselective C-5 (Het)Arylation of Mono- or Disubstituted Thiazolo[3,2-b][1,2,4]tri­azoles
[Full Papers]

Mikaël Le Meur, Stéphane Bourg, Stéphane Massip, Mathieu Marchivie, Christian Jarry, Gérald Guillaumet*, Sylvain Routier*

Coming soon.

Ruthenium-Catalyzed One-Pot Synthesis of (E)-(2-Arylvinyl)boronates through an Isomerization/Cross-Metathesis Sequence from Allyl-Substituted Aromatics
[Short Communications]

Rémy Hemelaere, Frédéric Caijo, Marc Mauduit, François Carreaux*, Bertrand Carboni

Published online on April 15, 2014.
DOI: 10.1002/ejoc.201402192

Synthesis of Di- and Trivalent Carbohydrate Mimetics with Oxepane Substructure by Employing Copper-Catalyzed [3+2] Cycloadditions of Alkynes with Azido­oxepanes
[Full Papers]

Léa Bouché, Hans-Ulrich Reissig*

Coming soon.

Neighboring ortho-Hydroxy Group Directed Catalytic Asymmetric Triple Domino Reactions of Acetaldehyde with (E)-2-(2-Nitrovinyl)phenols
[Short Communications]

Dhevalapally B. Ramachary*, P. Srinivasa Reddy, M. Shiva Prasad

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201402182

Cleavage of 2-(Arylamino)-4,6-dimethoxypyrimidines to Yield Arylguanidines
[Short Communications]

Julian W. Shaw, David H. Grayson, Isabel Rozas*

Coming soon.

A Three-Step Synthesis of the Guaianolide Ring System
[Short Communications]

Jan Hullaert, Duchan R. Laplace, Johan M. Winne*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201402170

Synthesis and Characterization of Bisumanenylidene
[Short Communications]

Toru Amaya, Takanori Ito, Toshikazu Hirao*

Coming soon.

Efficient Domino Synthesis of Pyrrole-Fused Isocoumarins with Microwave Heating
[Full Papers]

Mu-Yan Sun, Xiao-Yan Meng, Fu-Jie Zhao, Yi-Jing Dang, Fei Jiang, Kai Liu, Cong-Shuai Wang, Bo Jiang*, Shu-Jiang Tu*

Coming soon.

Acid-Catalyzed Domino Meinwald Rearrangement of Epoxides/Intramolecular [3+2] Cross-Cycloaddition of Cyclopropane-1,1-dicarboxylates
[Short Communications]

Wenju Zhu, Jun Ren, Zhongwen Wang*

Coming soon.

Synthesis of Trifluoromethyl-Substituted 3-Azabicyclo[n.1.0]alkanes: Advanced Building Blocks for Drug Discovery
[Full Papers]

Olexiy S. Artamonov, Evgeniy Y. Slobodyanyuk, Dmytro M. Volochnyuk, Igor V. Komarov, Andrey A. Tolmachev, Pavel K. Mykhailiuk*

Coming soon.

Disulfide Formation Strategies in Peptide Synthesis
[Microreviews]

Tobias M. Postma*, Fernando Albericio*

Coming soon.

Resorcin[4]arene-Based Molecular Baskets and Water-Soluble Container Molecules: Synthesis and 1H NMR Host–Guest Complexation Studies
[Full Papers]

Daniel Fankhauser, Dušan Kolarski, Wolfram R. Grüning, François Diederich*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402140

Palladium and TEMPO as Co-Catalysts in a Desulfinative Homocoupling Reaction
[Full Papers]

Dirk H. Ortgies, Fei Chen, Pat Forgione*

Coming soon.

Reactions of β-Azolylenamines with Sulfonyl Azides as an Approach to N-Unsubstituted 1,2,3-Triazoles and Ethene-1,2-diamines
[Full Papers]

Ilya Efimov, Vasiliy Bakulev*, Nikolai Beliaev, Tetyana Beryozkina, Uwe Knippschild, Johann Leban, Fan Zhi Zhin, Oleg Eltsov, Pavel Slepukhin, Marina Ezhikova, Wim Dehaen

Coming soon.

2,4- and 2,5-Disubstituted Arylthiazoles – Rapid Synthesis by C–H Coupling and Biological Evaluation
[Full Papers]

Lilia Lohrey, Takahiro N. Uehara, Satoshi Tani, Junichiro Yamaguchi*, Hans-Ulrich Humpf*, Kenichiro Itami*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201402129

Base-Catalyzed Domino Michael–Alkylation–Rearrangement Reaction: A Synthetic Route to Functionalized 2,3-Dihydrofurans
[Short Communications]

Ren-Zun Zhang, Chang-Yu Meng, Jian-Wu Xie*, Mei-Lan Xu, Wei-Dong Zhu*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201402126

Buchwald–Hartwig Amination Approach for the Synthesis of Functionalized 1,2,3,4-Tetrahydroacridine Derivatives
[Full Papers]

Julien de Sousa, Richard C. D. Brown, Rachid Baati*

Coming soon.

Combined Ugi-4CR/CuAAC Approach to Triazole-Based Neoglycolipids
[Full Papers]

Karell Pérez-Labrada, Ignacio Brouard*, Inmaculada Méndez, Carlos S. Pérez, José A. Gavín, Daniel G. Rivera*

Coming soon.

α-Acryloylamidoalkyl Sulfones in a Synthetic Approach for the Preparation of 6-Alkyltetrahydropyridin-2-ones
[Full Papers]

Nicola Lucchetti, Stefano Lancianesi, Marino Petrini*

Coming soon.

(+)-Sparteine-Mediated Substitution of o-Benzyl-N-pivaloylaniline with Ketones
[Full Papers]

Yi Kyung Ko, Chan Im, Junghwan Do, Yong Sun Park*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201402110

Synthesis of 1-(1H-Tetrazol-5-yl)-2H-iso­indole Derivatives through Ugi Four-Component and Silver-Catalyzed Reactions
[Full Papers]

Ran Wu, Shang Gao, Xu Chen, Guanghui Yang, Lingling Pan, Gaobo Hu, Ping Jia, Weihui Zhong, Chuanming Yu*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201402098

Synthesis and Absolute Configurations of Six Natural Phenylpropanoids
[Full Papers]

Xue-Lian Liu, Hui-Jun Chen, Yang-Yang Yang, Yikang Wu*, Jun You*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201402096

Palladium-Catalyzed Direct Arylation of Polyfluoroarenes with Organosilicon Reagents
[Short Communications]

Huixin Fan, Yaping Shang, Weiping Su*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402091

Straightforward Access to Hexahydropyrrolo[2,3-b]indole Core by a Regioselective C3-Azo Coupling Reaction of Arenediazonium Compounds with Tryptamines
[Full Papers]

David E. Stephens, Oleg V. Larionov*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402088

Fluorinated Sulfoximines: Preparation, Reactions and Applications
[Microreviews]

Xiao Shen, Jinbo Hu*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201402086

Biogenetically Inspired Total Synthesis of (+)-Liphagal: A Potent and Selective Phosphoinositide 3-Kinase α (PI3Kα) Inhibitor from the Marine Sponge Aka coralliphaga
[Full Papers]

Takaaki Kamishima, Takuya Kikuchi, Koichi Narita, Tadashi Katoh*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402082

Highly Stereoselective aza-Baylis–Hillman Reactions of CF3-Sulfinylimines: Straightforward Access to α-Methylene β-CF3 β-Amino Acids
[Short Communications]

Thierry Milcent*, Jing Hao, Kosuke Kawada, Vadim A. Soloshonok, Sandrine Ongeri, Benoit Crousse

Coming soon.

Solvent-Free Buchwald–Hartwig Reaction of Aryl and Heteroaryl Halides with Secondary Amines
[Short Communications]

Maxim A. Topchiy, Andrey F. Asachenko, Mikhail S. Nechaev*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402077

Enantioselective Fluorination of 2-Oxindoles by Structure-Micro-Tuned N-Fluorobenzenesulfonamides
[Full Papers]

Fajie Wang, Juli Li, Qingyang Hu, Xianjin Yang*, Xin-Yan Wu*, Haoming He

Coming soon.

Regioselective Synthesis of Highly Functionalized Furans Through the RuII-Catalyzed [3+2] Cycloaddition of Diazodi­carb­onyls
[Full Papers]

Likai Xia, Yong Rok Lee*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402067

Total Synthesis of Carbazomycin G by a Thermal Ring Expansion/Self-Redox Reaction Cascade
[Full Papers]

Yong An, Yunxia Wang, Xiangdong Hu*

Coming soon.

Asymmetric Diastereoselective Synthesis of Spirocyclopropane Derivatives of Oxindole
[Full Papers]

Maksim Ošeka, Artur Noole, Sergei Žari, Mario Öeren, Ivar Järving, Margus Lopp, Tõnis Kanger*

Coming soon.

Palladium-Catalyzed Allenylation/Intramolecular Diels–Alder Reaction of Furans with Propargyl Carboxylates for the Synthesis of Polycyclic Compounds
[Short Communications]

Chengyu Wang, Lingkai Kong, Yanli Li, Yanzhong Li*

Coming soon.

Regio-, and Stereoselective Iodobromination of Ynamides for Synthesis of (E)-1-Bromo-2-iodoenamides
[Full Papers]

Masataka Ide, Yuta Yauchi, Tetsuo Iwasawa*

Published online on April 9, 2014.
DOI: 10.1002/ejoc.201402057

Synthesis of Pyranonucleoside-6′-Triphosphates through the cycloSal-Method
[Full Papers]

Johanna Huchting, Chris Meier*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201402047

Transition-Metal-Free Approach to 4-Ethynylpyrimidines via Alkenynones
[Full Papers]

Pavel R. Golubev, Alena S. Pankova, Mikhail A. Kuznetsov*

Coming soon.

Catalyst-Free One-Pot Tandem Reduction of Oxo and Ene/Yne Functionalities by Hydrazine: Synthesis of Substituted Oxindoles­ from Isatins
[Short Communications]

Mukund Jha*, Ganesh M. Shelke, Anil Kumar

Published online on April 15, 2014.
DOI: 10.1002/ejoc.201402038

Gold(I)-, Palladium(II)-, Platinum(II)-, and Mercury(II)-Catalysed Spirocyclization of 1,3-Enynediols: Reaction Scope
[Full Papers]

Alexander Zhdanko*, Martin E. Maier*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201402029

Diterpenoid Alkaloid Lappaconine Derivative Catalyzed Asymmetric α-Hydroxylation of β-Dicarbonyl Compounds with Hydrogen Peroxide
[Full Papers]

Zhi Li, Mingming Lian, Fan Yang, Qingwei Meng*, Zhanxian Gao

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201402019

One-Pot Transformation of Methylarenes into Aromatic Aldehydes Under Metal-Free Conditions
[Full Papers]

Masayuki Tabata, Katsuhiko Moriyama, Hideo Togo*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201402015

Metal-Free Meerwein Carboarylation of Alkenes with Anilines: A Straightforward Approach to 3-Benzyl-3-alkyloxindoles
[Full Papers]

Dong Zhou, Ying-Chun Wang*, Shi Tang*

Coming soon.

Gold-Catalyzed 5-endo-dig Cyclization of 2-[(2-Aminophenyl)ethynyl]phenylamine with Ketones for the Synthesis of Spiroindolone and Indolo[3,2-c]quinolone Scaffolds
[Short Communications]

Basi. V. Subba Reddy*, Manisha Swain, S. Madhusudana Reddy, J. S. Yadav, B. Sridhar

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201402006

Copper-Catalyzed C(sp3)–C(sp2) Cross-Coupling: Synthesis of 4-Aryl-2-alkyl­amino-3-nitro-4H-chromenes
[Full Papers]

H. Surya Prakash Rao*, A. Veera Bhadra Rao

Coming soon.

Stereoselective Access to β-C-Glycosamines by Nitro-Michael Addition of Organolithium Reagents
[Short Communications]

Thierry Delaunay, Thomas Poisson*, Philippe Jubault, Xavier Pannecoucke*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201402001

One-Pot Glycosylations in the Synthesis of Human Milk Oligosaccharides
[Full Papers]

Camilla Arboe Jennum, Thomas Hauch Fenger, Linda M. Bruun, Robert Madsen*

Coming soon.

Unsymmetrical Bisphosphines for the Amidation of Aryl Chlorides: A Kinetic Study
[Full Papers]

Florian C. Falk, Peter Oechsle, Werner R. Thiel, Constantin-Gabriel Daniliuc, Jan Paradies*

Coming soon.

Copper(II)-Catalyzed Aromatization Followed by Bromination of Cyclohexenones Leading to Phenols and Bromophenols
[Full Papers]

Hung-Chun Tong, K. Rajender Reddy*, Shiuh-Tzung Liu*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201400158

Mechanistic Insight into the Lability of the Benzyloxycarbonyl (Z) Group in N-Protected Peptides under Mild Basic Conditions
[Full Papers]

Marta Tena-Solsona, César A. Angulo-Pachón, Beatriu Escuder*, Juan F. Miravet*

Coming soon.

Sulfur–Carbon Bond Formation through Ring-Opening of Triazolothiadiazole with Organometallics
[Full Papers]

Raja Ben Othman, Stéphane Massip, Mathieu Marchivie, Christian Jarry, Johnny Vercouillie, Sylvie Chalon, Gérald Guillaumet, Franck Suzenet*, Sylvain Routier*

Published online on April 8, 2014.
DOI: 10.1002/ejoc.201400151

Stereocontrolled Synthesis of the C1–C10 Building Block (“Southwestern Moiety”) for the Unnatural Enantiomers of the Polyene Polyol Antibiotics Filipin III and Pentamycin. A Sultone Forming Ring-Closing Metathesis for Protection of Homoallylic Alcohols
[Full Papers]

Patrick Walleser, Reinhard Brückner*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201400145

syn/anti Switching by Specific Heteroatom–Titanium Coordination in the Mannich-Like Synthesis of 2,3-Diaryl-β-amino Acid Derivatives
[Full Papers]

Andrea Bonetti, Francesca Clerici, Francesca Foschi, Donatella Nava, Sara Pellegrino, Michele Penso*, Raffaella Soave, Maria Luisa Gelmi*

Published online on April 8, 2014.
DOI: 10.1002/ejoc.201400142

Palladium-Catalyzed Suzuki Cross-Cou­pling of Phenylhydrazine or (Phenylsulfonyl)hydrazine
[Short Communications]

Yahui Li, Wei Liu, Qingshan Tian, Qing Yang, Chunxiang Kuang*

Published online on April 15, 2014.
DOI: 10.1002/ejoc.201400126

Synthesis and Selected Reactivity Studies of a Dissymmetric (Phosphinoylmethylpyridine N-Oxide) Methylamine Platform
[Full Papers]

Sabrina Ouizem, Sylvie L. Pailloux, Alisha D. Ray, Eileen N. Duesler, Diane A. Dickie, Robert T. Paine*, Benjamin P. Hay

Published online on April 8, 2014.
DOI: 10.1002/ejoc.201400120

Arylethynyl-Substituted Tristriazolotriazines – Synthesis, Optical Properties, and Thermotropic Behavior
[Full Papers]

Stefan Glang, Thorsten Rieth, Dorothee Borchmann, Ilaria Fortunati, Raffaella Signorini, Heiner Detert*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201400088

Regioselective O2′,O3′-Deacetylations of Peracetylated Ribonucleosides by Using Tetra-n-butylammonium Fluoride
[Short Communications]

Arun Babu Kumar, Roman Manetsch*

Coming soon.

Sulfoximine-Based Modular Enantioselective Synthesis of Azaspirocycles Featuring Sulfoximine Displacement, Dianion Cycloalkylation, RCM and N-Acyliminium Ion Formation
[Full Papers]

Adeline Köhler (née Adrien), Gerhard Raabe, Jan Runsink, Franz Köhler, Hans-Joachim Gais*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201400068

BODIPY Fluorophore Toolkit for Probing Chemical Reactivity and for Tagging Reactive Functional Groups
[Full Papers]

Eva M. Hensle, N. Melody Esfandiari, Sung-Gon Lim, Suzanne A. Blum*

Coming soon.

Iron-Catalyzed Oxidative 1,2-Carboacylation of Activated Alkenes with Alcohols: A Tandem Route to 3-(2-Oxoethyl)indolin-2-ones
[Full Papers]

Xuan-Hui Ouyang, Ren-Jie Song*, Jin-Heng Li*

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201400043

Ligand-Free Ullmann-Type C–Heteroatom Couplings Under Practical Conditions
[Full Papers]

Imma Güell, Xavi Ribas*

Published online on April 14, 2014.
DOI: 10.1002/ejoc.201400033

Regioselective Hydrodebromination of ­Polybrominated Indoles
[Full Papers]

Giorgio Chelucci*, Gérard A. Pinna, Giansalvo Pinna

Coming soon.

Domino Recombinant γ-Isomerization and Reverse Wacker Oxidation of γ-Vinyl-γ-butyro­lactone: Synthesis of (+)-trans-, (–)- and (+)-Disparlures
[Full Papers]

Venkati Bethi, Pullaiah Kattanguru, Rodney A. Fernandes*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201400021

Syntheses of Functionalized Allylamines via Lithiated Intermediates
[Full Papers]

Samia Firdous, Uli Kazmaier*

Published online on April 8, 2014.
DOI: 10.1002/ejoc.201400017

Copper-Catalyzed Intramolecular Oxidative C(sp3)–H Amidation of 2-Aminoacetophenones: Efficient Synthesis of Indoline-2,3-diones
[Short Communications]

Jinbo Huang*, Tingting Mao, Qiang Zhu*

Published online on April 10, 2014.
DOI: 10.1002/ejoc.201400012

One-Pot Stereoselective Synthesis of (Z)-β-Ketoenamides from β-Halo α,β-Unsaturated Aldehydes
[Full Papers]

Junali Gogoi, Pranjal Gogoi*, Romesh C. Boruah*

Coming soon.

Synthesis of Phenyl-1-benzoxepinols Isolated from Butcher's Broom and Analogous Benzoxepines
[Full Papers]

Josef M. Herrmann, Monika Untergehrer, Guido Jürgenliemk, Jörg Heilmann*, Burkhard König*

Published online on April 8, 2014.
DOI: 10.1002/ejoc.201400004

Synthesis of 1,2,3-Triazoles from Azide-Derivatised Aminocyclitols by Catalytic Diazo Transfer and CuAAC Click Chemistry
[Full Papers]

Li Ji, Guo-Quan Zhou, Chao Qian*, Xin-Zhi Chen

Published online on April 17, 2014.
DOI: 10.1002/ejoc.201301874

Di- and Tricationic Organic Salts: An Overview of Their Properties and Applications
[Microreviews]

Francesca D'Anna, Renato Noto*

Published online on April 11, 2014.
DOI: 10.1002/ejoc.201301871

Regioselective Biomimetic Oxidative ­Cyclization Strategy for the Synthesis of Aryldihydronaphthalene Lignans
[Full Papers]

Wenling Li*, Hao Liu, Jingyan Xu, Peng Zang, Qian Liu, Wenbo Li

Published online on April 15, 2014.
DOI: 10.1002/ejoc.201301825

[8+2] Formal Cycloaddition Reactions of Tropones with Azlactones under Brønsted Acid Catalysis and Synthesis of α-(2-Tropyl), α-Alkyl α-Amino Acids
[Full Papers]

Francisco Esteban, Ricardo Alfaro, Francisco Yuste, Alejandro Parra, José Luis García Ruano*, José Alemán*

Coming soon.

Design and Synthesis of a Monofluoro-Substituted Aromatic Amino Acid as a Conformationally Restricted 19F NMR ­Label for Membrane-Bound Peptides
[Full Papers]

Anton N. Tkachenko, Pavel K. Mykhailiuk*, Dmytro S. Radchenko, Oleg Babii, Sergii Afonin*, Anne S. Ulrich*, Igor V. Komarov

Coming soon.

Long-Range Diastereoselectivity in an Ugi Reaction: Stereocontrolled and Diversity-Oriented Synthesis of Tetrahydrobenz­oxazepines
[Full Papers]

Luca Banfi*, Alessandro Bagno, Andrea Basso, Carlo De Santis, Renata Riva, Federico Rastrelli

Coming soon.

Synthesis of Atorvastatin Lactone Linker Constructs for Target Fishing
[Full Papers]

Pramod Sawant, Martin E. Maier*

Coming soon.

Visible-Light-Triggered Direct Benzoyloxy­lation of Electron-Rich Arenes at Room Temperature without Chelation Assistance
[Short Communications]

Honghua Rao, Ping Wang, Chao-Jun Li*

Coming soon.

Synthesis and Stability Studies of α,α-Difluoro Ester Phospholipids
[Full Papers]

Palle J. Pedersen, Thomas L. Andresen, Mads H. Clausen*

Coming soon.

Diaryl-Substituted Perylenetetracarboxdi­imides: Synthesis, Separation, Characteri­zation and Comparison of Electrochemical and Optical Properties of 1,7- and 1,6-Regioisomer
[Full Papers]

Somnath Dey*, Alexander Efimov, Helge Lemmetyinen

Coming soon.

The 1-Phenyl-1-Trimethylsilyl Ethyl Cation: An NMR Spectroscopic and Computational Study of the α-Silyl Effect in Benzyl Cations
[Full Papers]

Arseni Kostenko, Bernhard Müller, Frank-Peter Kaufmann, Yitzhak Apeloig*, Hans-Ullrich Siehl*

Coming soon.

Synthesis of Naturally Occurring Cyclohexene Rings Using Stereodirected Intramolecular Diels–Alder Reactions Through Asymmetric 1,3-Dioxane Tethering
[Full Papers]

Hajer Abdelkafi, Laurent Evanno, Alexandre Deville, Lionel Dubost, Angèle Chiaroni, Bastien Nay*

Coming soon.

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