European Journal of Organic Chemistry

Cover image for Vol. 2014 Issue 31

Editor: Haymo Ross, Deputy Editor: Susan Wilkinson

Impact Factor: 3.154

ISI Journal Citation Reports © Ranking: 2013: 14/58 (Chemistry Organic)

Online ISSN: 1099-0690

Associated Title(s): Advanced Synthesis & Catalysis, Asian Journal of Organic Chemistry

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Here's a selection of upcoming papers. Also see the EarlyView page for the latest papers published online.

Transition-Metal-Free Oxidative Iodination of 1,3,4-Oxadiazoles
[Short Communications]

Carl Albrecht Dannenberg, Vincent Bizet, Liang-Hua Zou, Carsten Bolm*

Coming soon.

High-Temperature Synthesis of Amides from Alcohols or Aldehydes by Using Flow Chemistry
[Short Communications]

Nida Ambreen, Thomas Wirth*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403280

Practical Access to Aromatic Thiocyanates by CuCN-Mediated Direct Aerobic Oxidative Cyanation of Thiophenols and Diaryl Disulfides
[Short Communications]

Thomas Castanheiro, Mihaela Gulea*, Morgan Donnard*, Jean Suffert*

Coming soon.

The First Bidirectional [4+2] Cycloadditions of Benzo[1,2:4,5]dicyclobutenes: Synthesis of Benzo[1,2-f:4,5-f′]diisoindole-1,3,7,9-tetraones
[Full Papers]

Ismail Abdelshafy Abdelhamid, Holger Butenschön*

Coming soon.

Nickel-Catalyzed Decarboxylative Arylation of Heteroarenes through sp2 C–H Functionalization
[Short Communications]

Ke Yang, Peng Wang, Cheng Zhang, Adnan A. Kadi, Hoong-Kun Fun, Yan Zhang*, Hongjian Lu*

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201403234

Iron(II)-Catalyzed Asymmetric Epoxidation of Trisubstituted α,β-Unsaturated ­Esters
[Short Communications]

Lan Luo, Hisashi Yamamoto*

Coming soon.

An Economical and Practical Synthesis of rac-(Z)-β-Santalol: Application of a ­Scriabine-Inspired Reaction to Alkenes ­Results in the One-Step Preparation of a Key Intermediate
[Short Communications]

Anthony A. Birkbeck*, Xavier Marquet, Pascal Millet, Hervé Pamingle

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403219

Room-Temperature Direct Alkenylation of 3-Arylsydnones
[Short Communications]

Yiwen Yang*, Chunxiang Kuang*

Coming soon.

Stereoselective Synthesis of Highly Substituted α-Silylamines from Silylmethyl Azides under Ru Catalysis
[Short Communications]

Wook Jeong, Jungjoon Kim, Jaiwook Park*, Young Ho Rhee*

Published online on October 22, 2014.
DOI: 10.1002/ejoc.201403200

Total Synthesis of (±)-Oxalicumone C and Chiral Resolution and Elucidation of its Absolute Configuration
[Short Communications]

Christoph Wink, Lars Andernach, Till Opatz, Siegfried R. Waldvogel*

Coming soon.

Rapid Synthesis of Unsymmetrical Sulfo­rhodamines through Nucleophilic Amination of a Monobrominated Sulfoxanthene Dye
[Full Papers]

Arnaud Chevalier, Kevin Renault, Frédéric Boschetti, Pierre-Yves Renard*, Anthony Romieu*

Coming soon.

Enantioselective Synthesis of Spiroimines by Asymmetric Decarboxylative Alkyl­ation/Isomerization/[3+2]-Cycloaddition Reaction of Azidoalkenes
[Full Papers]

Matt Rambla, Leslie Duroure, Laurent Chabaud*, Catherine Guillou*

Published online on October 24, 2014.
DOI: 10.1002/ejoc.201403161

Nonsymmetrical Azocarbonamide Carb­oxylates as Effective Mitsunobu Reagents
[Short Communications]

Daniel P. Furkert*, Benjamin Breitenbach, Ludovic Juen, Ina Sroka, Mathilde Pantin, Margaret A. Brimble*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403152

Palladium-Catalyzed Decarboxylative Methylthiolation of Aromatic Carboxylic Acids by Using DMSO as the Sulfurizing Reagent
[Short Communications]

Zhengjiang Fu, Zhaojie Li, Qiheng Xiong, Hu Cai*

Coming soon.

Mechanistic Elucidation of the 2-Nor­bornyl to 1,3-Dimethylcyclopentenyl Cation Isomerization
[Full Papers]

Said Jalife, Gerardo Martínez-Guajardo, Claudia Zavala-Oseguera, María A. Fernández-Herrera*, Paul von Rague Schleyer*, Gabriel Merino*

Published online on October 27, 2014.
DOI: 10.1002/ejoc.201403146

Triphosgene-Mediated Couplings in the Solid Phase: Total Synthesis of Brachystemin A
[Short Communications]

Lijing Fang, Chunlei Wu, Zaidan Yu, Peng Shang, Yongxian Cheng, Yuefeng Peng*, Wu Su*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403145

Design and Synthesis of 3-Trifluoromethyl-3H-pyrazoles and Further Investigations of Their Transformation to 1H-Pyrazoles
[Full Papers]

Qiang Sha, Haixuan Liu, and Yunyang Wei*

Published online on October 27, 2014.
DOI: 10.1002/ejoc.201403141

Synthesis of Vicinal Diketoses by Using a Metathesis–Hydroxylation–Oxidation Sequence
[Full Papers]

Melchior Menzel, Thomas Ziegler*

Published online on October 24, 2014.
DOI: 10.1002/ejoc.201403140

Role of Side-Chain Bioisosteres in Determining the Binding Affinity of Click Chemistry Derived RGD Peptidomimetics to αvβ3 Integrin
[Full Papers]

Pierangelo Fabbrizzi*, Gloria Menchi, Silvia Raspanti, Antonio Guarna, Andrea Trabocchi*

Published online on October 24, 2014.
DOI: 10.1002/ejoc.201403129

Protecting-Group-Free Diastereoselective Total Synthesis of (±)-6-epi-Cleistenolide and Chemoenzymatic Synthesis of (–)-6-epi-Cleistenolide
[Full Papers]

Pankaj S. Mahajan, Rajesh G. Gonnade, Santosh B. Mhaske*

Coming soon.

Comparison of Linear and Cross-Conjugation from Rates of Vinylheptafulvene Ring-Closure
[Full Papers]

Kasper Fjelbye, Trine Nørgaard Christensen, Martyn Jevric, Søren Lindbæk Broman, Anne Ugleholdt Petersen, Anders Kadziola, Mogens Brøndsted Nielsen*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403117

Stereoselective Synthesis of α-Trifluoro­methyl Enones by AuI/CuI-Co-Catalyzed Tandem 1,3-Acyloxy Migration/Trifluoro­methylation Reaction of Propargyl Acetates
[Full Papers]

Yun-Long Ji, Jin-Hong Lin*, Ji-Chang Xiao*, Yu-Cheng Gu

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403115

Cationic Trialkylphosphates: Synthesis and Transfection Efficacies Compared to Phosphoramidate Analogues
[Full Papers]

Stéphanie S. Le Corre, Mathieu Berchel, Tony Le Gall, Jean-Pierre Haelters, Pierre Lehn, Tristan Montier, Paul-Alain Jaffrès*

Coming soon.

Synthesis and NMR Analysis of 1,4-Disubstituted 1,2,3-Triazoles Tethered to Pyr­idine, Pyrimidine, and Pyrazine Rings
[Full Papers]

Aljoša Bolje, Damijana Urankar, Janez Košmrlj*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201403100

Iron-Catalyzed [4C+1N] Cyclization of 4-Acetylenic Ketones with Primary Amines: Synthesis of 5-(Aryl)alkylidene-4,5-dihydropyrroles
[Short Communications]

Bo Sun, Quan Ma, Yeming Wang, Yuegang Zhao, Peiqiu Liao, Xihe Bi*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403097

Enantioselective Allylation of tert-Butyldimethylsilyl-Protected Vanillin and Synthesis of a Lignan Derivative Isolated from Machilus wangchiana
[Short Communications]

Timothée Cadart, Petr Koukal, Martin Kotora*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403094

Design of a Ribosyltriazole-Annulated Cyclooctyne for Oligonucleotide Labeling by Strain-Promoted Alkyne–Azide Cycloaddition
[Short Communications]

Pieter van Delft, Wilbert de Witte, Nico J. Meeuwenoord, Gerbrand J. van der Heden van Noort, Frank Versluis, Rene C. L. Olsthoorn, Herman S. Overkleeft, Gijs A. van der Marel*, Dmitri V. Filippov*

Published online on October 22, 2014.
DOI: 10.1002/ejoc.201403086

Rhodium(III)-Catalyzed One-Pot Access to Isoquinolines and Heterocycle-Fused Pyrid­ines in Aqueous Medium through C–H Cleavage
[Full Papers]

Jitan Zhang, Hongsheng Qian, Zhanxiang Liu, Chunhua Xiong*, Yuhong Zhang*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201403085

Prins–Arylthiolation Reaction on Terpenoids: Diastereoselective Synthesis of 4-Arylthiooctahydro-2H-chromenes
[Short Communications]

Barnali Sarmah, Gakul Baishya*, Rajani K. Baruah

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403080

Stereocontrolled Construction of the 3,4-Dihydrothiacarbazol-2(9H)-one Skeleton by Using Bifunctional Squaramide-Catalyzed Cascade Reactions
[Full Papers]

Shanren Chen, Jianping Pan, Youming Wang, Zhenghong Zhou*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201403078

Synthesis of All Eight Stereoisomeric 6-Deoxy-l-hexopyranosyl Donors – Trends in Using Stereoselective Reductions or Mitsunobu Epimerizations
[Full Papers]

Tobias Gylling Frihed, Christian Marcus Pedersen*, Mikael Bols

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403074

Asymmetric Synthesis of 3,4-Disubstituted Proline Derivatives: Application in Synthesis of Hepatitis C Virus Protease Inhibitor Telaprevir
[Full Papers]

Fan Zhang, Xiaoan Wen, Qing-Long Xu*, Hongbin Sun*

Coming soon.

Copper-Catalyzed Regioselective Cross-Dehydrogenative Coupling of Coumarins with Benzylic Csp3–H Bonds
[Full Papers]

Shi-Liu Zhou, Li-Na Guo, Xin-Hua Duan*

Coming soon.

Stereoselective Synthesis of C-2-Methylene and C-2-Methyl α- and β-C-Glycosides from 2-C-Branched Glycals: Formal Total Synthesis of (–)-Brevisamide
[Full Papers]

Chalapala Sudharani, Patteti Venukumar, Perali Ramu Sridhar*

Coming soon.

A Versatile Protocol for the Synthesis of Pyrazolyl-Substituted Pyridinium and Guanidinium Salts from Pyridone and Urea Derivatives
[Full Papers]

Antje K. C. Echterhoff, Jutta Kösters, Roland Fischer, Jan J. Weigand*

Published online on October 27, 2014.
DOI: 10.1002/ejoc.201403057

DNA Recognition with Polycyclic-Aromatic-Hydrocarbon-Presenting Calixarene Conjugates
[Full Papers]

Antonio Rescifina*, Chiara Zagni, Placido G. Mineo, Salvatore V. Giofrè, Ugo Chiacchio, Stefano Tommasone, Carmen Talotta, Carmine Gaeta, Placido Neri*

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201403050

A Palladium Catalyst Supported on Carb­on-Coated Cobalt Nanoparticles – Preparation of Palladium-Free Biaryls by Suzuki–Miyaura Reactions in Ethanol
[Full Papers]

Antoine Derible, Carine Diebold, Joseph Dentzer, Roger Gadiou, Jean-Michel Becht*, Claude Le Drian*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403038

Enzyme-Catalyzed Kinetic Resolution of 2,2,2-Trifluoro-1-(heteroaryl)ethanols: Experimental and Docking Studies
[Full Papers]

Olexandr V. Kucher, Anastasiya O. Kolodiazhnaya, Oleg B. Smolii, Dmytro V. Prisuazhnyk, Katerina A. Tolmacheva, Yurii S. Moroz*, Pavel K. Mykhailiuk*, Andrey A. Tolmachev

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201403013

Recent Advances in Stereoselective [2+2+2] Cycloadditions
[Microreviews]

Muriel Amatore*, Corinne Aubert

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201403012

Highly Efficient Synthesis of Allenes from Trimethylaluminum Reagent and Propargyl Acetates Mediated by a Palladium Catalyst
[Full Papers]

Qing-Han Li*, Jung-Yuan Jeng, Han-Mou Gau*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201403008

Synthesis of Isotopically Labelled Oligo­prenyl Diphosphates and Their Application in Mechanistic Investigations of Terpene Cyclases
[Full Papers]

Christian A. Citron, Patrick Rabe, Lena Barra, Chiaki Nakano, Tsutomu Hoshino, Jeroen S. Dickschat*

Published online on October 24, 2014.
DOI: 10.1002/ejoc.201403002

Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condensation to Isoxazolo[60]fullerenes
[Full Papers]

Giacomo Biagiotti, Stefano Cicchi, Francesco De Sarlo, and Fabrizio Machetti*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201402990

Syntheses of Chiral Ferrocenophanes and Their Application to Asymmetric Catalysis
[Short Communications]

Qiying Zhang, Xiuling Cui*, Lianmei Chen, Haitao Liu, Yangjie Wu*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201402985

Biosynthetically Distinct Cytotoxic Polyketides from Setophoma terrestris
[Full Papers]

Tamam El-Elimat, Mario Figueroa, Huzefa A. Raja, Tyler N. Graf, Steven M. Swanson, Joseph O. Falkinham III, Mansukh C. Wani, Cedric J. Pearce, Nicholas H. Oberlies*

Coming soon.

Construction and Multiple Exterior Surface Functionalization of Giant Molecular Cages
[Full Papers]

Muhammad Moazzam Naseer, De-Xian Wang, Liang Zhao, Mei-Xiang Wang*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201402963

Ruthenium-Catalyzed Alkenylation of ­Arenes with Alkynes or Alkenes by 1,2,3-Triazole-Directed C–H Activation
[Full Papers]

Xing Guang Li, Kai Liu, Gang Zou, Pei Nian Liu*

Published online on October 29, 2014.
DOI: 10.1002/ejoc.201402938

Efficient Cross-Coupling of Dioxazaborocanes with α-Phosphate Enamides
[Full Papers]

Nicolas Gigant*, Aurélien Honraedt, Emmanuel Gras*, Isabelle Gillaizeau*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201402927

Synthetic Strategies for the Synthesis and Transformation of Substituted Pyrrolinones as Advanced Intermediates for Rhazinilam Analogues
[Full Papers]

Inga Kholod, Olivier Vallat, Ana-Maria Buciumas, Antonia Neels, and Reinhard Neier*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201402903

Synthesis of Galactoclusters by Metal-Free Thiol “Click Chemistry” and Their Binding Affinities for Pseudomonas aeruginosa Lectin LecA
[Full Papers]

Caroline Ligeour, Lucie Dupin, Alberto Marra, Gérard Vergoten, Albert Meyer, Alessandro Dondoni, Eliane Souteyrand, Jean-Jacques Vasseur, Yann Chevolot*, François Morvan*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201402902

SNH- and SNipso-Arylamination of 1,3,7-Triazapyrenes
[Full Papers]

Ivan Borovlev*, Oleg Demidov, Nadezhda Saigakova, Gulminat Amangasieva

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201402891

Chiral Squaramide-Catalyzed Sulfa-Michael/Aldol Cascade for the Asymmetric Synthesis of Spirocyclic Tetrahydrothiophene Chromanone Derivatives
[Full Papers]

Bo-Liang Zhao, Lei Liu, Da-Ming Du*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201402889

Convenient Synthesis of the Antibiotic Linez­olid via an Oxazolidine-2,4-dione Intermediate Derived from the Chiral Building Block Isoserine
[Full Papers]

Arianna Greco, Rossella De Marco, Sara Tani, Daria Giacomini, Paola Galletti, Alessandra Tolomelli, Eusebio Juaristi, Luca Gentilucci*

Published online on October 28, 2014.
DOI: 10.1002/ejoc.201402888

Iron(III)-Catalyzed C–H Functionalization: ortho-Benzoyloxylation of N,N-Dialkylanilines and its Application to 1,4-Benzoxazepines
[Full Papers]

Barreddi Chiranjeevi, BotlaVinayak, Thupakula Parsharamulu, Vemulapalli S. PhaniBabu, Bharatam Jagadeesh, Balasubramanian Sridhar, Malapaka Chandrasekharam*

Published online on October 30, 2014.
DOI: 10.1002/ejoc.201402751

A Synthetic Route to Sulfobetaine Methacrylates with Varying Charge Distance
[Full Papers]

Domenic Kratzer, Leonie Barner, Christian Friedmann, Stefan Bräse, Joerg Lahann*

Coming soon.

Synthesis and Structural Characterization of 2:1 [α/Aza]-oligomers
[Full Papers]

Zhou Zhou, Cheng Deng, Cécile Abbas, Claude Didierjean, Marie-Christine Averlant-Petit*, Jacques Bodiguel, Régis Vanderesse, Brigitte Jamart-Grégoire*

Published online on October 21, 2014.
DOI: 10.1002/ejoc.201402628

A Robust and Efficient Catalyst Possessing an Electron-Deficient Ligand for the Palladium-Catalyzed Direct Arylation of Heteroarenes
[Short Communications]

Alexandra Jakab, Zoltán Dalicsek, Tibor Soós*

Coming soon.

[8+2] Formal Cycloaddition Reactions of Tropones with Azlactones under Brønsted Acid Catalysis and Synthesis of α-(2-Tropyl), α-Alkyl α-Amino Acids
[Full Papers]

Francisco Esteban, Ricardo Alfaro, Francisco Yuste, Alejandro Parra, José Luis García Ruano*, José Alemán*

Coming soon.

Long-Range Diastereoselectivity in an Ugi Reaction: Stereocontrolled and Diversity-Oriented Synthesis of Tetrahydrobenz­oxazepines
[Full Papers]

Luca Banfi*, Alessandro Bagno, Andrea Basso, Carlo De Santis, Renata Riva, Federico Rastrelli

Coming soon.

Synthesis of Atorvastatin Lactone Linker Constructs for Target Fishing
[Full Papers]

Pramod Sawant, Martin E. Maier*

Coming soon.

Visible-Light-Triggered Direct Benzoyloxy­lation of Electron-Rich Arenes at Room Temperature without Chelation Assistance
[Short Communications]

Honghua Rao, Ping Wang, Chao-Jun Li*

Coming soon.

Synthesis and Stability Studies of α,α-Difluoro Ester Phospholipids
[Full Papers]

Palle J. Pedersen, Thomas L. Andresen, Mads H. Clausen*

Coming soon.

Diaryl-Substituted Perylenetetracarboxdi­imides: Synthesis, Separation, Characteri­zation and Comparison of Electrochemical and Optical Properties of 1,7- and 1,6-Regioisomer
[Full Papers]

Somnath Dey*, Alexander Efimov, Helge Lemmetyinen

Coming soon.

The 1-Phenyl-1-Trimethylsilyl Ethyl Cation: An NMR Spectroscopic and Computational Study of the α-Silyl Effect in Benzyl Cations
[Full Papers]

Arseni Kostenko, Bernhard Müller, Frank-Peter Kaufmann, Yitzhak Apeloig*, Hans-Ullrich Siehl*

Coming soon.

Synthesis of Naturally Occurring Cyclohexene Rings Using Stereodirected Intramolecular Diels–Alder Reactions Through Asymmetric 1,3-Dioxane Tethering
[Full Papers]

Hajer Abdelkafi, Laurent Evanno, Alexandre Deville, Lionel Dubost, Angèle Chiaroni, Bastien Nay*

Coming soon.

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