ChemMedChem

Preview

Here's a selection of upcoming papers. Also see the EarlyView page for the latest papers published online.

Structure–Activity Relationship Analysis of the Peptide Deformylase Inhibitor 5-Bromo-1H-indole-3-acetohydroxamic Acid
[Full Paper]

Sylvain Petit, Yann Duroc, Valéry Larue, Carmela Giglione, Carole Léon, Coralie Soulama, Alexis Denis, Frédéric Dardel, Thierry Meinnel, Isabelle Artaud*

Coming soon.

Synthesis of an ¹¹C-Labeled Antiprion GN8 Derivative and Evaluation of Its Brain Uptake by Positron Emission Tomography
[Communication]

Tsutomu Kimura, Takeo Sako, Siqin, Junji Hosokawa-Muto, Yi Long Cui, Yasuhiro Wada, Yosky Kataoka, Hisashi Doi, Suehiro Sakaguchi, Masaaki Suzuki, Yasuyoshi Watanabe, Kazuo Kuwata*

Published online on May 24, 2013.
DOI: 10.1002/cmdc.201300167

Probing the Structural Properties of DNA/RNA Grooves with Sterically Restricted Phosphonium Dyes: Screening of Dye Cytotoxicity and Uptake
[Full Paper]

Ivo Crnolatac, Lidija-Marija Tumir, Nedyalko Y. Lesev, Aleksey A. Vasilev, Todor G. Deligeorgiev, Katarina Mišković, Ljubica Glavaš-Obrovac, Oliver Vugrek, Ivo Piantanida*

Coming soon.

Modification of Triclosan Scaffold in Search of Improved Inhibitors for Enoyl-Acyl Carrier Protein (ACP) Reductase in Toxoplasma gondii
[Full Paper]

Jozef Stec, Alina Fomovska, Gustavo A. Afanador, Stephen P. Muench, Ying Zhou, Bo-Shiun Lai, Kamal El Bissati, Mark R. Hickman, Patty J. Lee, Susan E. Leed, Jennifer M. Auschwitz, Caroline Sommervile, Stuart Woods, Craig W. Roberts, David Rice, Sean T. Prigge, Rima McLeod*, Alan P. Kozikowski*

Coming soon.