ChemMedChem

Cover image for Vol. 11 Issue 3

Editor-in-Chief: Natalia Ortúzar

Impact Factor: 2.968

ISI Journal Citation Reports © Ranking: 2014: 19/59 (Chemistry Medicinal); 83/255 (Pharmacology & Pharmacy)

Online ISSN: 1860-7187

Associated Title(s): Angewandte Chemie International Edition, Chemistry - A European Journal, Chemistry – An Asian Journal, ChemBioChem, Medicinal Research Reviews, Molecular Informatics

Preview

Here's a selection of upcoming papers. Also see the EarlyView page for the latest papers published online.

Antivirulence Isoquinolone Mannosides: Optimization of the Biaryl Aglycone for FimH Lectin Binding Affinity and Efficacy in the Treatment of Chronic UTI
[Communication]

Cassie Jarvis, Zhenfu Han, Vasilios Kalas, Roger Klein, Jerome S. Pinkner, Bradley Ford, Jana Binkley, Corinne K. Cusumano, Zachary Cusumano, Laurel Mydock-McGrane, Scott J. Hultgren*, James W. Janetka*

Published online on February 5, 2016.
DOI: 10.1002/cmdc.201600006

Fragment Screening of Soluble Epoxide Hydrolase for Lead Generation—Structure-Based Hit Evaluation and Chemistry Exploration
[Full Paper]

Yafeng Xue*, Thomas Olsson, Carina A Johansson, Linda Öster, Hans-Georg Beisel, Mattias Rohman, David Karis, Stefan Bäckström

Published online on February 4, 2016.
DOI: 10.1002/cmdc.201500575

Substrate Activity Screening (SAS) and Related Approaches in Medicinal Chemistry
[Minireview]

Rafaela Gladysz, Anne-Marie Lambeir, Jurgen Joossens, Koen Augustyns, Pieter Van der Veken*

Published online on February 4, 2016.
DOI: 10.1002/cmdc.201500569

Cancer Immunotherapy: Selected Targets and Small-Molecule Modulators
[Review]

Hilmar Weinmann*

Published online on February 2, 2016.
DOI: 10.1002/cmdc.201500566

A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression
[Communication]

Stefano Guglielmo*, Marialessandra Contino, Loretta Lazzarato, Maria Grazia Perrone, Marco Blangetti, Roberta Fruttero, Nicola Antonio Colabufo*

Published online on February 2, 2016.
DOI: 10.1002/cmdc.201500538

Current Experimental Methods for Characterizing Protein–Protein Interactions
[Review]

Mi Zhou, Qing Li, Renxiao Wang*

Coming soon.

Serpin A1 C-Terminal Peptides as Collagen Turnover Modulators
[Full Paper]

Simona Pascarella, Caterina Tiberi, Giuseppina Sabatino, Francesca Nuti, Anna Maria Papini, Lisa Giovannelli*, Paolo Rovero*

Coming soon.

Structural Re-engineering of the α-Helix Mimetic JY-1-106 into Small Molecules: Disruption of the Mcl-1–Bak-BH3 Protein–Protein Interaction with 2,6-Di-Substituted Nicotinates
[Communication]

Brandon Drennen, Jacob A. Scheenstra, Jeremy L. Yap, Lijia Chen, Maryanna E. Lanning, Braden M. Roth, Paul T. Wilder, Steven Fletcher*

Published online on February 4, 2016.
DOI: 10.1002/cmdc.201500461

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