ChemMedChem

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Here's a selection of upcoming papers. Also see the EarlyView page for the latest papers published online.

Structure–Activity Relationship Analysis of the Peptide Deformylase Inhibitor 5-Bromo-1H-indole-3-acetohydroxamic Acid
[Full Paper]

Sylvain Petit, Yann Duroc, Valéry Larue, Carmela Giglione, Carole Léon, Coralie Soulama, Alexis Denis, Frédéric Dardel, Thierry Meinnel, Isabelle Artaud*

Coming soon.

Conjugates of Cisplatin and Cyclooxygenase Inhibitors as Potent Antitumor Agents Overcoming Cisplatin Resistance
[Communication]

Wilma Neumann, Brenda C. Crews, Lawrence J. Marnett, Evamarie Hey-Hawkins*

Coming soon.

Mechanistic and Cytotoxicity Studies of Group IV β-Diketonate Complexes
[Communication]

Rianne M. Lord, James J. Mannion, Andrew J. Hebden, Adi E. Nako, Benjamin D. Crossley, Max W. McMullon, Felix D. Janeway, Roger M. Phillips, Patrick C. McGowan*

Coming soon.

Photodelivery of CO by Designed PhotoCORMs: Correlation between Absorption in the Visible Region and Metal–CO Bond Labilization in Carbonyl Complexes
[Full Paper]

Indranil Chakraborty, Samantha J. Carrington, Pradip K. Mascharak*

Published online on April 23, 2014.
DOI: 10.1002/cmdc.201402007

Photoinduced Intercalation and Coordination of a Dirhodium Complex to DNA: Dual DNA Binding
[Full Paper]

Alycia M. Palmer, Scott J. Burya, Judith C. Gallucci, Claudia Turro*

Published online on April 17, 2014.
DOI: 10.1002/cmdc.201402004

Insight into the Recognition, Binding, and Reactivity of Catalytic Metallodrugs Targeting Stem Loop IIb of Hepatitis C IRES RNA
[Full Paper]

Seth S. Bradford, Martin James Ross, Insiya Fidai, J. A. Cowan*

Published online on April 22, 2014.
DOI: 10.1002/cmdc.201400070

Getting to the Source: Selective Drug Targeting of Cancer Stem Cells
[Minireview]

Fatima Ismail, David A. Winkler*

Published online on April 23, 2014.
DOI: 10.1002/cmdc.201400068

Development of 3-Phenyl-N-(2-(3-phenylureido)ethyl)-thiophene-2-sulfonamide Compounds as Inhibitors of Antiapoptotic Bcl-2 Family Proteins
[Full Paper]

Chengwen Yang, Sha Chen, Mi Zhou, Yan Li, Yangfeng Li, Zhengxi Zhang, Zhen Liu, Qian Ba, Jingquan Li, Hui Wang, Xiaomei Yang*, Dawei Ma*, Renxiao Wang*

Coming soon.

Investigation of a Vitamin B12 Conjugate as a PET Imaging Probe
[Full Paper]

Oluwatayo F. Ikotun, Bernadette V. Marquez, Christopher H. Fazen, Anna R. Kahkoska, Robert P. Doyle*, Suzanne E. Lapi*

Published online on April 17, 2014.
DOI: 10.1002/cmdc.201400048

Discovery of 14-3-3 Protein–Protein Interaction Inhibitors that Sensitize Multidrug-Resistant Cancer Cells to Doxorubicin and the Akt Inhibitor GSK690693
[Full Paper]

Mattia Mori, Giulia Vignaroli, Ylenia Cau, Jelena Dinić, Richard Hill, Matteo Rossi, David Colecchia, Milica Pešić, Wolfgang Link, Mario Chiariello, Christian Ottmann, Maurizio Botta*

Coming soon.

Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2-Amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6H-quinazolin-5-one Oxime
[Full Paper]

Raffaella Amici*, Chiara Bigogno, Roberto Boggio, Andrea Colombo, Stephen M. Courtney, Roberto Dal Zuffo, Giulio Dondio, Fulvia Fusar, Stefania Gagliardi, Saverio Minucci, Marco Molteni, Christian A. G. N. Montalbetti, Annalisa Mortoni, Mario Varasi, Stefania Vultaggio, Ciro Mercurio

Published online on April 17, 2014.
DOI: 10.1002/cmdc.201400037

Design, Synthesis, and Activity Evaluation of GK/PPARγ Dual-Target-Directed Ligands as Hypoglycemic Agents
[Communication]

Jianxun Lu, Lei Lei, Yi Huan, Yongqiang Li, Lijing Zhang, Zhufang Shen, Wenxiang Hu, Zhiqiang Feng*

Published online on April 15, 2014.
DOI: 10.1002/cmdc.201400009

Unfolding and Conformational Variations of Thrombin-Binding DNA Aptamers: Synthesis, Circular Dichroism and Molecular Dynamics Simulations
[Full Paper]

Lidan Sun, Hongwei Jin, Xiaoyang Zhao, Zhenming Liu, Yifu Guan, Zhenjun Yang, Liangren Zhang*, Lihe Zhang

Coming soon.

Insight into the Functional and Structural Properties of 3-Arylcoumarin as an Interesting Scaffold in Monoamine Oxidase B Inhibition
[Full Paper]

Maria João Matos*, Santiago Vilar, Verónica García-Morales, Nicholas P. Tatonetti, Eugenio Uriarte, Lourdes Santana, Dolores Viña

Published online on April 17, 2014.
DOI: 10.1002/cmdc.201300533

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