Cover image for Vol. 11 Issue 18

Editorial Board Chairs: Antonello Mai, Rainer Metternich. Assoc. Editors: David Peralta, Scott Williams (Sr)

Impact Factor: 2.98

ISI Journal Citation Reports © Ranking: 2015: 18/59 (Chemistry Medicinal); 76/253 (Pharmacology & Pharmacy)

Online ISSN: 1860-7187

Associated Title(s): Angewandte Chemie International Edition, Chemistry - A European Journal, Chemistry – An Asian Journal, ChemBioChem, Medicinal Research Reviews, Molecular Informatics

March 07, 2013

Articles by the ChemMedChem Board

Articles by the ChemMedChem BoardMembers of the ChemMedChem Editorial (EB) and International Advisory (IAB) Boards are key to the direction and continued success our journal. They set the standard of quality both in peer review and by submitting their own contributions for publication. Below is a list of articles our Board members have authored or co-authored over the past year alone. We extend our continued gratitude to everyone on the EB and IAB for helping shape and maintain the high quality of ChemMedChem's content.

Christopher Abell (IAB):

Discovery of Schaeffer's Acid Analogues as Lead Structures of Mycobacterium tuberculosis Type II Dehydroquinase Using a Rational Drug Design Approach

Maurizio Botta (EB):

Synthesis, Biological Activity, and ADME Properties of Novel S-DABOs/N-DABOs as HIV Reverse Transcriptase Inhibitors

A Combination Strategy to Inhibit Pim-1: Synergism between Noncompetitive and ATP-Competitive Inhibitors

Computational Studies Identifying Entry Inhibitor Scaffolds Targeting the Phe43 Cavity of HIV-1 gp120

Maria José Camarasa (IAB):

Dipeptidyl Peptidase IV (DPPIV/CD26)-Based Prodrugs of Hydroxy-Containing Drugs

Dipeptidyl Peptidase IV-Activated Prodrugs of Anti-Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems

Paul Coleman (IAB):

Discovery of [(2R,5R)-5-{[(5-Fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl][5-methyl-2-(pyrimidin-2-yl)phenyl]methanone (MK-6096): A Dual Orexin Receptor Antagonist with Potent Sleep-Promoting Properties

Paul Coleman (IAB) and Steven Young (EB):

Editorial: Challenges and Opportunities in Neuroscience Research

François Diederich (IAB):

Identification of 1,3-Diiminoisoindoline Carbohydrazides as Potential Antimalarial Candidates

Efficient Stacking on Protein Amide Fragments

Beat Ernst (IAB):

From a Library of MAG Antagonists to Nanomolar CD22 Ligands

FimH Antagonists: Structure–Activity and Structure–Property Relationships for Biphenyl a-D-Mannopyranosides

Alpine Drug Discovery Summit: 10th Swiss Course on Medicinal Chemistry

Concepción González-Bello (IAB):

Comparative Binding Energy (COMBINE) Analysis for Understanding the Binding Determinants of Type II Dehydroquinase Inhibitors

Stephen Hanessian (IAB):

Crystal Structures of a Bioactive 6'-Hydroxy Variant of Sisomicin Bound to the Bacterial and Protozoal Ribosomal Decoding Sites

Adriaan P. IJzerman (IAB):

Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E-4031 Analogues

Substructure-Based Virtual Screening for Adenosine A2A Receptor Ligands

Hualiang Jiang (IAB):

Recent Advances in Neuraminidase Inhibitor Development as Anti-influenza Drugs

Gerhard Klebe (EB) and Rolf Müller (IAB):

Development of Improved PPARβ/δ Inhibitors

Gerhard Klebe (EB):

Experimental and Computational Active Site Mapping as a Starting Point to Fragment-Based Lead Discovery

Water Makes the Difference: Rearrangement of Water Solvation Layer Triggers Non-additivity of Functional Group Contributions in Protein–Ligand Binding

Beyond Heparinization: Design of Highly Potent Thrombin Inhibitors Suitable for Surface Coupling

Novel Type II Fatty Acid Biosynthesis (FAS II) Inhibitors as Multistage Antimalarial Agents

Alan P. Kozikowski (IAB):

Chiral Mercaptoacetamides Display Enantioselective Inhibition of Histone Deacetylase 6 and Exhibit Neuroprotection in Cortical Neuron Models of Oxidative Stress

Ulf Madsen (IAB):

Structure–Activity Relationships for Negative Allosteric mGluR5 Modulators

Marco Mor (IAB):

Structure–Activity Relationships and Mechanism of Action of Eph–ephrin Antagonists: Interaction of Cholanic Acid with the EphA2 Receptor

Marco Mor (IAB) and Giorgio Tarzia (EB):

MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-{[(3-O-Substituted)anilino]alkyl}amides

Klaus Müller (IAB) and Martin Stahl (EB):

Design of Libraries Targeting Protein–Protein Interfaces

Tudor I. Oprea (IAB):

A Chemogenomic Analysis of Ionization Constants—Implications for Drug Discovery

Thomas Ryckmans (IAB):

Application of Barluenga Boronic Coupling (BBC) to the Parallel Synthesis of Drug-like and Drug Fragment-like Molecules

Carlo Scolastico (IAB):

Synthesis of Gd and 68Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor-Imaging Probes

Henning Steinhagen (IAB):

Editorial: Channeling Drug Discovery

Paul Wyatt (IAB):

Design, Synthesis and Biological Evaluation of Trypanosoma brucei Trypanothione Synthetase Inhibitors

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